SCHEMBL10651297

SCHEMBL10651297

COC(=O)c1cc2cc(S)ccc2oc1=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.67
ALDH1A1 P00352 5/20 0.67
CA12 O43570 4/20 0.67
CA2 P00918 4/20 0.67
CA6 P23280 4/20 0.67
CA7 P43166 4/20 0.67
CA9 Q16790 4/20 0.67
CA14 Q9ULX7 4/20 0.67
CA5B Q9Y2D0 4/20 0.67
HPGD P15428 3/20 0.67
CA3 P07451 3/20 0.67
CA5A P35218 3/20 0.67
ATM Q13315 1/20 0.55
MAOB P27338 10/20 0.55
CA1 P00915 2/20 0.52
MAOA P21397 2/20 0.52
GAA P10253 1/20 0.52
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
CA4 P22748 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17903545 0.84 MAOB (0.72) KDM4EALDH1A1CA12CA2CA6
SCHEMBL29985431 0.84 KDM4E (0.68) KDM4EALDH1A1CA12CA2CA6
SCHEMBL18589240 0.84 MAOB (0.70) KDM4EALDH1A1CA12CA2CA6
SCHEMBL6835643 0.82 KDM4E (0.76) KDM4EALDH1A1CA12CA2CA6
SCHEMBL22502678 0.82 MEN1 (0.72) KDM4EALDH1A1CA12CA2CA6
SCHEMBL1808756 0.82 MAOA (0.71) KDM4EALDH1A1CA12CA2CA6
SCHEMBL29575367 0.81 CA12 (0.65) KDM4EALDH1A1CA12CA2CA6
SCHEMBL18752472 0.81 CA12 (0.82) KDM4EALDH1A1CA12CA2CA6
SCHEMBL76086 0.80 KDM4E (1.00) KDM4EALDH1A1CA12CA2CA6
SCHEMBL5858940 0.80 LMNA (0.47) KDM4EALDH1A1CA12CA2CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0123543-B1 LEUKOTRIENE ANTAGONISTS, THEIR PRODUCTION AND USE AND COMPOSITIONS CONTAINING THEM MERCK FROSST CANADA INC. (CA) 1988-02-03 EP disclosed
US-4609744-A 4-oxo-benzopyran carboxylic acids MERCK FROSST CANADA INC. (CA) 1986-09-02 US disclosed
EP-0123543-A1 Leukotriene antagonists, their production and use and compositions containing them MERCK FROSST CANADA INC. (CA) 1984-10-31 EP disclosed