SCHEMBL10653259

SCHEMBL10653259

O=C(O)CN1C(=S)CSc2ccc(F)cc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
CYP1A2 P05177 2/20 0.39
HSD17B10 Q99714 1/20 0.39
ALDH1A1 P00352 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
NOTUM Q6P988 1/20 0.38
TP53 P04637 4/20 0.36
HSD17B3 P37058 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
TSHR P16473 1/20 0.36
MAPT P10636 4/20 0.35
LMNA P02545 1/20 0.35
KDM4E B2RXH2 1/20 0.34
CYP2D6 P10635 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10652752 0.89 HSD17B3 (0.44) MEN1KMT2AGSK3AGSK3BCYP1A2
SCHEMBL10649933 0.85 ALDH1A1 (0.48) MEN1KMT2AGSK3AGSK3BALDH1A1
SCHEMBL30808596 0.85 ALDH1A1 (0.48) MEN1KMT2AGSK3AGSK3BALDH1A1
SCHEMBL10511618 0.84 LMNA (0.45) MEN1KMT2AGSK3AGSK3BCYP1A2
SCHEMBL10511348 0.83 FPR2 (0.48) MEN1KMT2AGSK3AGSK3BCYP1A2
SCHEMBL10507993 0.81 HSD17B10 (0.44) MEN1KMT2AHSD17B10ALDH1A1CYP3A4
SCHEMBL4971828 0.80 NPSR1 (0.48) MEN1KMT2AGSK3AGSK3BCYP1A2
SCHEMBL10509865 0.78 MEN1 (0.42) MEN1KMT2AGSK3AGSK3BCYP1A2
SCHEMBL10509886 0.76 HSD17B3 (0.44) MEN1KMT2AGSK3AGSK3BCYP1A2
SCHEMBL10511482 0.75 CHRM2 (0.45) MEN1KMT2ACYP1A2ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4755509-A Heterocyclic aldose reductase inhibitors and methods of using them Carbipem (FR) 1988-07-05 US disclosed