SCHEMBL10511348

SCHEMBL10511348

O=C(O)CN1C(=S)CSc2ccc(C(F)(F)F)cc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 4/20 0.48
HSD17B3 P37058 1/20 0.47
ALDH1A1 P00352 1/20 0.46
PKM P14618 1/20 0.46
RAD52 P43351 1/20 0.41
AR P10275 1/20 0.40
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
HDAC6 Q9UBN7 2/20 0.39
HTT P42858 1/20 0.39
GAA P10253 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10511510 0.86 ALDH1A1 (0.56) FPR2HSD17B3ALDH1A1PKMRAD52
SCHEMBL10650608 0.84 NPSR1 (0.50) FPR2HSD17B3ALDH1A1PKMRAD52
SCHEMBL10653259 0.83 MEN1 (0.40) HSD17B3ALDH1A1HPGDMEN1KMT2A
SCHEMBL10511618 0.81 LMNA (0.45) HSD17B3ALDH1A1NPSR1MEN1KMT2A
SCHEMBL10507726 0.78 KCNN4 (0.39) FPR2HSD17B3MEN1KMT2AGAA
SCHEMBL10507993 0.78 HSD17B10 (0.44) HSD17B3ALDH1A1HPGDNPSR1MEN1
SCHEMBL4971828 0.77 NPSR1 (0.48) HSD17B3ALDH1A1NPSR1MEN1KMT2A
SCHEMBL30808641 0.77 ALDH1A1 (0.47) FPR2HSD17B3ALDH1A1PKMRAD52
SCHEMBL11037157 0.76 FPR2 (0.45) FPR2HSD17B3ALDH1A1PKMRAD52
SCHEMBL11037153 0.76 FPR2 (0.45) FPR2HSD17B3ALDH1A1PKMRAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0162776-B1 HETEROCYCLIC DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS USEFUL AS ALDOSE REDUCTASE INHIBITORS CONTAINING THEM LABORATOIRES UPSA (FR) 1989-04-19 EP disclosed
US-4755509-A Heterocyclic aldose reductase inhibitors and methods of using them Carbipem (FR) 1988-07-05 US disclosed
EP-0162776-A2 Heterocyclic derivatives, process for their preparation and medicaments useful as aldose reductase inhibitors containing them LABORATOIRES UPSA (FR) 1985-11-27 EP disclosed