SCHEMBL10656178

SCHEMBL10656178

O=C(c1ccccc1)C(Br)CF

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 1/20 0.47
TDP1 Q9NUW8 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CES1 P23141 7/20 0.45
CES2 O00748 5/20 0.45
LMNA P02545 1/20 0.45
GSK3B P49841 2/20 0.43
PTPN1 P18031 1/20 0.43
ALKBH5 Q6P6C2 1/20 0.43
PGR P06401 1/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
HTR2A P28223 1/20 0.43
HRH1 P35367 1/20 0.43
KCNH2 Q12809 1/20 0.43
KMT2A Q03164 2/20 0.42
MAPK1 P28482 3/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3730123 0.80 CES2 (0.54) L3MBTL1CES1CES2LMNAKMT2A
SCHEMBL6455139 0.79 MDM2 (0.47) MDM2TDP1L3MBTL1CES1CES2
SCHEMBL2336670 0.79 PGR (0.52) MDM2TDP1L3MBTL1CES1CES2
SCHEMBL5054802 0.79 ALKBH5 (0.47) MDM2TDP1L3MBTL1CES1CES2
SCHEMBL10658190 0.79 MAPK1 (0.48) MDM2TDP1L3MBTL1CES1CES2
SCHEMBL10658140 0.79 CES1 (0.44) MDM2TDP1L3MBTL1CES1CES2
SCHEMBL5214256 0.78 GSK3B (0.47) MDM2TDP1L3MBTL1CES1CES2
SCHEMBL4257686 0.78 MDM2 (0.66) MDM2TDP1L3MBTL1CES1CES2
SCHEMBL8780874 0.77 CES1 (0.52) MDM2TDP1L3MBTL1CES1CES2
SCHEMBL18705724 0.77 MDM2 (0.48) MDM2TDP1L3MBTL1CES1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0167945-B1 PHENYLETHYLAMINOPROPIOPHENONE DERIVATIVES, PROCESS FOR THEIR PREPARATION ET MEDICINES CONTAINING THEM Troponwerke GmbH & Co. KG (DE) 1988-04-13 EP disclosed
EP-0167945-A2 Phenylethylaminopropiophenone derivatives, process for their preparation et medicines containing them Troponwerke GmbH & Co. KG (DE) 1986-01-15 EP disclosed