SCHEMBL1065677

SCHEMBL1065677

Cc1onc(-c2c(F)cccc2Cl)c1C(=O)Cl

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.68
SMN1; SMN2 Q16637 3/20 0.68
KMT2A Q03164 3/20 0.67
GPBAR1 Q8TDU6 1/20 0.65
ATM Q13315 3/20 0.64
MEN1 O00255 1/20 0.64
GLA P06280 1/20 0.64
HPGD P15428 1/20 0.64
HTT P42858 1/20 0.64
ALDH1A1 P00352 3/20 0.63
TSHR P16473 1/20 0.62
POLB P06746 2/20 0.61
ALOX15 P16050 1/20 0.61
GAA P10253 2/20 0.60
NPC1 O15118 1/20 0.60
MAPT P10636 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30881266 1.00 LMNA (0.68) LMNASMN1; SMN2KMT2AGPBAR1ATM
SCHEMBL6644159 0.91 LMNA (0.56) LMNASMN1; SMN2KMT2AGPBAR1ATM
SCHEMBL3451560 0.90 TSHR (0.75) LMNASMN1; SMN2KMT2AGPBAR1MEN1
SCHEMBL899628 0.89 LMNA (0.68) LMNASMN1; SMN2KMT2AGPBAR1ATM
SCHEMBL10520781 0.89 LMNA (0.68) LMNASMN1; SMN2KMT2AGPBAR1ATM
SCHEMBL7184918 0.88 TSHR (0.82) LMNASMN1; SMN2KMT2AGPBAR1ATM
SCHEMBL10332625 0.88 LMNA (0.67) LMNASMN1; SMN2KMT2AGPBAR1ATM
Anthranilic Acid SCHEMBL7870197 0.87 LMNA (0.62) LMNASMN1; SMN2KMT2AGPBAR1ATM
SCHEMBL11893412 0.85 ALDH1A1 (0.72) LMNASMN1; SMN2KMT2AGPBAR1ATM
SCHEMBL14519854 0.85 KMT2A (0.67) LMNASMN1; SMN2KMT2AGPBAR1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 147 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102964356-A Synthesis method of flucloxacillin sodium HEZE RUIZHI TECHNOLOGY DEV CO LTD 2013-03-13 CN claimed
CN-102702227-A Preparation method for flucloxacillin sodium HEBEI HUARI PHARMACEUTICAL CO LTD 2012-10-03 CN claimed
US-20040010005-A1 Stereoselective process for preparing cylcohexyl amine derivatives BARNETT CHARLES JACKSON (US) 2004-01-15 US claimed
EP-1322652-A1 STEREOSELECTIVE PROCESS FOR PREPARING CYCLOHEXYL AMINE DERIVATIVES ELI LILLY AND COMPANY (US) 2003-07-02 EP claimed
WO-2002024705-A1 STEREOSELECTIVE PROCESS FOR PREPARING CYCLOHEXYL AMINE DERIVATIVES ELI LILLY AND COMPANY (US) 2002-03-28 WO claimed
CN-117964622-A Novel isoxazole compound and preparation method and application thereof 河北科技大学 2024-05-03 CN disclosed
CN-115819228-A Synthetic method of 2-aryl-2-cyclohexanedione enol ester compound 南方医科大学 2023-03-21 CN disclosed
EP-4074708-A1 1-(4-(ISOXAZOL-5-YL)-1H-PYRAZOL-1-YL)-2-METHYLPROPAN-2-OL DERIVATIVES AND RELATED COMPOUNDS AS IL-7 AND IFN-GAMMA INHIBITORS FOR TREATING AUTOIMMUNE DISEASES AND CHRONIC INFLAMMATION Immunic AG (DE) 2022-10-19 EP disclosed
EP-3679034-B1 1-(4-(ISOXAZOL-5-YL)-1H-PYRAZOL-1-YL)-2-METHYLPROPAN-2-OL DERIVATIVES AND RELATED COMPOUNDS AS IL-7 AND IFN-GAMMA INHIBITORS FOR TREATING AUTOIMMUNE DISEASES AND CHRONIC INFLAMMATION IMMUNIC AG (DE) 2022-06-01 EP disclosed
US-11292788-B2 IL-17 and IFN-gamma inhibition for the treatment of autoimmune diseases and chronic inflammation IMMUNIC AG (DE) 2022-04-05 US disclosed
CN-109400630-B Synthetic method of flucloxacillin sodium 浙江普洛得邦制药有限公司 2021-07-02 CN disclosed
US-20210061796-A1 IL-17 and IFN-gamma inhibition for the treatment of autoimmune diseases and chronic inflammation IMMUNIC AG (DE) 2021-03-04 US disclosed
EP-1067928-A1 METHODS FOR INHIBITING MRP1 ELI LILLY AND COMPANY (US) 2001-01-17 EP disclosed
WO-1999051236-A1 METHODS FOR INHIBITING MRP1 ELI LILLY AND COMPANY (US) 1999-10-14 WO disclosed
WO-1999051227-A1 METHODS FOR INHIBITING MRP1 ELI LILLY AND COMPANY (US) 1999-10-14 WO disclosed
WO-1999051228-A1 METHODS FOR INHIBITING MRP1 ELI LILLY AND COMPANY (US) 1999-10-14 WO disclosed
EP-0265185-A2 Cephalosporins, processes for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1988-04-27 EP disclosed
US-4179511-A Antibacterial 3-(5-tetrazolyl) penam compounds PFIZER INC. (US) 1979-12-18 US disclosed
US-4143039-A ANTIBACTERIAL 3-(5-TETRAZOLYL)PENAM COMPOUNDS PFIZER INC. (US) 1979-03-06 US disclosed
US-4115385-A PENICILLINS PFIZER INC. (US) 1978-09-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210061796-A1 IL-17 and IFN-gamma inhibition for the treatment of autoimmune diseases and chronic inflammation IFNG, IL17A, IFNAR1 LMNA 3556/4885SMN1; SMN2 4231/4885KMT2A 1459/4885
US-20040010005-A1 Stereoselective process for preparing cylcohexyl amine derivatives ALKBH3, AZI2, ALKBH1 LMNA 864/4885SMN1; SMN2 2439/4885KMT2A 411/4885
US-11292788-B2 IL-17 and IFN-gamma inhibition for the treatment of autoimmune diseases and chronic inflammation IFNG, IL17A, IFNAR1 LMNA 3556/4885SMN1; SMN2 4231/4885KMT2A 1459/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.