SCHEMBL1067702

SCHEMBL1067702

COc1cc(NC(=O)[C@H](CCSC(F)(F)F)NC(=O)O)cc(OC)c1OC

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP2C9 P11712 1/20 0.44
ALDH1A1 P00352 2/20 0.43
MMP2 P08253 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
METAP2 P50579 1/20 0.40
HTT P42858 1/20 0.39
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TSHR P16473 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1068136 0.88 CYP1A2 (0.49) CYP2C19CYP2C9MMP2MEN1KMT2A
SCHEMBL12933711 0.87 ABCB1 (0.43) CYP3A4CYP2C19CYP2C9ALDH1A1MMP2
SCHEMBL12933684 0.83 CYP3A4 (0.49) CYP3A4CYP2C19CYP2C9ALDH1A1MEN1
Hydrochloric Acid SCHEMBL2787536 0.82 CYP3A4 (0.48) CYP3A4CYP2C19CYP2C9ALDH1A1MEN1
Hydrochloric Acid SCHEMBL2787531 0.82 CYP3A4 (0.48) CYP3A4CYP2C19CYP2C9ALDH1A1MEN1
SCHEMBL12933712 0.76 ALDH1A1 (0.49) CYP2C19CYP2C9ALDH1A1MMP2MEN1
SCHEMBL1066478 0.74 MAPK1 (0.46) ALDH1A1KMT2A
SCHEMBL12933704 0.74 MAPK1 (0.46) ALDH1A1KMT2A
SCHEMBL5470679 0.73 CA12 (0.46) ALDH1A1MMP2L3MBTL1
SCHEMBL12933681 0.70 CYP1A2 (0.55) CYP2C19CYP2C9SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7868206-B2 Trihalomethionine derivative and pharmaceutical product containing the same National University Corporation, Gunma University (JP) 2011-01-11 US disclosed
US-20100076224-A1 NOVEL TRIHALOMETHIONINE DERIVATIVE AND PHARMACEUTICAL PRODUCT CONTAINING THE SAME NATIONAL UNIVERSITY CORPORATION GUNMA UNIVERSITY (JP) 2010-03-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100076224-A1 NOVEL TRIHALOMETHIONINE DERIVATIVE AND PHARMACEUTICAL PRODUCT CONTAINING THE SAME CTH, MTR, BHMT CYP3A4 262/4885CYP2C19 472/4885CYP2C9 367/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.