SCHEMBL10691127

SCHEMBL10691127

Cc1cn2ccc3c(Cl)cccc3c2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.42
CYP2A6 P11509 3/20 0.42
ALDH1A1 P00352 3/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 1/20 0.40
NR4A2 P43354 2/20 0.37
PDE10A Q9Y233 2/20 0.36
TYMS P04818 1/20 0.35
NOTUM Q6P988 1/20 0.34
ADRA2A P08913 1/20 0.34
KDM4E B2RXH2 3/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
MAPT P10636 2/20 0.34
PKM P14618 1/20 0.34
GRM5 P41594 1/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
NFKB1 P19838 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10426160 0.78 PDE10A (0.56) ALDH1A1HPGDHSD17B10PDE10AKDM4E
SCHEMBL3256643 0.76 ALDH1A1 (0.54) CYP1A2CYP2A6ALDH1A1HPGDHSD17B10
SCHEMBL11250574 0.75 ALDH1A3 (0.52) ALDH1A1HPGDHSD17B10KDM4ENPC1
SCHEMBL8563007 0.73 ADRA2B (0.37) CYP1A2KDM4ENPC1RAB9AMAPT
SCHEMBL8563013 0.72 DOT1L (0.35) ALDH1A1HPGDHSD17B10PDE10AKDM4E
SCHEMBL8561058 0.72 CYP3A4 (0.42) CYP1A2PDE10AKDM4ENPC1RAB9A
SCHEMBL10694973 0.71 MAPK1 (0.47) CYP1A2MAPTGRM5MEN1KMT2A
SCHEMBL10691749 0.71 POLB (0.40) ALDH1A1HPGDNR4A2KDM4ENPC1
SCHEMBL10692077 0.71 CYP1A2 (0.42) CYP1A2CYP2A6ALDH1A1NR4A2PDE10A
SCHEMBL20085840 0.70 ALDH1A1 (0.38) ALDH1A1HPGDHSD17B10PDE10AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4738967-A Imidazoisoquinoline compounds useful as anti-ulcerative agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-04-19 US disclosed
US-4686227-A Imidazoisoquinoline compounds useful as anti-ulcerative agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-08-11 US disclosed
EP-0165545-A2 Imidazoisoquinoline compounds and processes for preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1985-12-27 EP disclosed