SCHEMBL10691826

SCHEMBL10691826

CN1C(=O)C(C)(c2ccccc2OCCCCN2CCN(CCCC(c3ccc(F)cc3)c3ccc(F)cc3)CC2)Cc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.43
ADRA1A P35348 6/20 0.43
HRH1 P35367 6/20 0.43
DRD3 P35462 6/20 0.43
OPRK1 P41145 6/20 0.43
SLC6A3 Q01959 6/20 0.43
LMNA P02545 5/20 0.43
OPRM1 P35372 5/20 0.43
HTR6 P50406 5/20 0.43
CACNA1C Q13936 5/20 0.43
ADORA3 P0DMS8 5/20 0.43
OPRD1 P41143 5/20 0.43
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
HTR2C P28335 4/20 0.43
DRD2 P14416 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
CYP3A4 P08684 4/20 0.43
CYP2D6 P10635 4/20 0.43
KCNH2 Q12809 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL10754715 0.94 HTR2A (0.41) HTR2AADRA1AHRH1DRD3OPRK1
SCHEMBL10694474 0.88 CYP3A4 (0.41) HTR2AADRA1AHRH1DRD3OPRK1
SCHEMBL10759482 0.87 SLC6A3 (0.42) HTR2AADRA1AHRH1DRD3OPRK1
Hydrochloric Acid SCHEMBL10692827 0.86 SLC6A3 (0.42) HTR2AADRA1AHRH1DRD3OPRK1
Hydrochloric Acid SCHEMBL10409299 0.83 LMNA (0.43) HTR2AADRA1AHRH1DRD3OPRK1
Hydrochloric Acid SCHEMBL10695977 0.77 DRD2 (0.42) HTR2AADRA1ADRD3DRD2TDP1
Hydrochloric Acid SCHEMBL10570034 0.75 MEN1 (0.38) HTR2AADRA1AHRH1DRD3OPRK1
SCHEMBL10689170 0.71 ADRA1A (0.40) ADRA1ADRD3MEN1KMT2ADRD2
Hydrochloric Acid SCHEMBL10770827 0.71 MEN1 (0.35) HTR2AADRA1AHRH1DRD3OPRK1
Hydrochloric Acid SCHEMBL10573477 0.70 ABCB1 (0.39) HTR2AADRA1AHRH1DRD3OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed