SCHEMBL10691956

SCHEMBL10691956

COc1cncc2sc(-c3ccccc3)c(OC)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
FYN P06241 1/20 0.38
GAK O14976 1/20 0.37
MAP3K8 P41279 1/20 0.37
EGFR P00533 1/20 0.36
ICAM1 P05362 1/20 0.36
SELE P16581 1/20 0.36
VCAM1 P19320 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
BRAF P15056 1/20 0.36
TUBB4A P04350 2/20 0.36
TUBB P07437 2/20 0.36
TUBA3C P0DPH7 2/20 0.36
TUBA1B P68363 2/20 0.36
TUBA4A P68366 2/20 0.36
TUBB4B P68371 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28238880 0.67 FYN (0.60) KDM4EALDH1A1HPGDCTDSP1FYN
SCHEMBL16763232 0.65 PDE4A (0.35) KDM4EALDH1A1HPGDTUBB4ATUBB
SCHEMBL9869471 0.64 BRAF (0.37) KDM4EALDH1A1HPGDCTDSP1EGFR
SCHEMBL11331212 0.64 KDM4E (0.40) KDM4EALDH1A1HPGDFYNEGFR
SCHEMBL10744711 0.64 HSP90AA1 (0.44) KDM4EALDH1A1HPGDMAPK1KMT2A
SCHEMBL11521411 0.63 HSD17B1 (0.48) KDM4EALDH1A1HPGDFYNEGFR
SCHEMBL4396043 0.62 ACHE (0.48) KDM4EALDH1A1HPGDFYNBRAF
Methoxy Aucuparin SCHEMBL8420787 0.62 KDM4E (0.62) KDM4EALDH1A1HPGDCTDSP1FYN
Dimethylamine SCHEMBL619459 0.62 FYN (0.50) KDM4EALDH1A1HPGDCTDSP1FYN
SCHEMBL28338665 0.61 HPGD (0.61) KDM4EALDH1A1HPGDCTDSP1FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4767766-A Derivatives of 3-hydroxyazabenzo(B)thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-08-30 US disclosed