SCHEMBL9869471

SCHEMBL9869471

COCOc1c(-c2ccccc2)sc2cnccc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
CASP1 P29466 1/20 0.36
HTT P42858 1/20 0.36
CASP7 P55210 1/20 0.36
NCOA1 Q15788 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RCE1 Q9Y256 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
LIMK1 P53667 1/20 0.34
HSP90AA1 P07900 1/20 0.34
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
ALOX5 P09917 1/20 0.33
ESR1 P03372 1/20 0.32
KDM4C Q9H3R0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9868772 0.76 ALOX5 (0.46) BRAFKDM4EALDH1A1GLAGAA
SCHEMBL9869116 0.76 KDM4E (0.43) KDM4EALDH1A1GAAHPGD
SCHEMBL657642 0.71 BRAF (0.42) BRAFKDM4EALDH1A1GLAGAA
SCHEMBL9868855 0.71 ALOX5 (0.45) BRAFKDM4EALDH1A1GLAGAA
SCHEMBL5620698 0.71 ALDH1A1 (0.46) BRAFKDM4EALDH1A1GLAGAA
SCHEMBL9869316 0.70 LMNA (0.40) KDM4ENCOA3
SCHEMBL9869324 0.69 HSPA5 (0.31)
SCHEMBL9870113 0.66 CNR1 (0.45) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9869497 0.66 ALOX5 (0.46) KDM4EGAAHTTHSD17B10ALOX5
SCHEMBL10691956 0.64 KDM4E (0.39) BRAFKDM4EALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5026941-A Catalytic alkylation of naphthalene and/or 2-isopropyl-naphthalene in the presence of a saturated polycarbocyclic compound to yield 2,6- and 2,7-diisopropylnaphthalene TOSHO CORPORATION (JP) 1991-06-25 US disclosed
US-5006532-A Enzyme inhibitor; antiinflammatory agents MERCK & CO. INC., INC. (US) 1991-04-09 US disclosed
US-4904672-A Derivatives of 3-hydroxyazabenzo[b]thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1990-02-27 US disclosed
US-4767766-A Derivatives of 3-hydroxyazabenzo(B)thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-08-30 US disclosed