SCHEMBL10692521

SCHEMBL10692521

C=CCOc1c(NC(C)=O)c[c]cc1OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
PKM P14618 1/20 0.40
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
DRD1 P21728 1/20 0.38
HTR2A P28223 1/20 0.38
PTGS1 P23219 2/20 0.38
PTGS2 P35354 2/20 0.38
ALDH1A1 P00352 4/20 0.37
HTT P42858 2/20 0.37
GABRA1 P14867 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37
GABRB2 P47870 1/20 0.37
NPC1 O15118 1/20 0.37
HSP90AA1 P07900 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
MAPT P10636 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5597577 0.81 ALDH1A1 (0.42) KDM4EALDH1A1HTTMAPTCYP1A2
SCHEMBL15666382 0.76 LIG1 (0.40) KDM4EPOLBSMN1; SMN2HTR2AALDH1A1
SCHEMBL3551171 0.72 CYP3A4 (0.40) KDM4EPOLBSMN1; SMN2PTGS1PTGS2
SCHEMBL3959073 0.69 FLT3 (0.54) PKMALDH1A1NPC1HPGDRAB9A
SCHEMBL10631908 0.69 BRD4 (0.61) KDM4EPOLBSMN1; SMN2ALDH1A1NPC1
SCHEMBL30428722 0.69 BRD4 (0.61) KDM4EPOLBSMN1; SMN2ALDH1A1NPC1
SCHEMBL5888949 0.68 HPGD (0.37) SMN1; SMN2HTR2APTGS1PTGS2ALDH1A1
SCHEMBL1355596 0.66 ALDH1A1 (0.45) KDM4ESMN1; SMN2ALDH1A1HTTNPC1
SCHEMBL7771748 0.66 HSD17B1 (0.46) PKMSMN1; SMN2ALDH1A1MAPTGAA
SCHEMBL9024109 0.64 LMNA (0.45) KDM4EPOLBSMN1; SMN2PTGS2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4757084-A Pharmaceuticals MERCK & CO., INC. (US) 1988-07-12 US disclosed
EP-0217204-A1 Trans-2-(3,4,5-trimethoxyphenyl)-5-(5,6-dimethoxy-3-pyridyl)-tetrahydrothiophene, a PAF-antagonist MERCK & CO. INC. (US) 1987-04-08 EP disclosed