SCHEMBL5597577

SCHEMBL5597577

COc1c[c]cc(NC(C)=O)c1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 1/20 0.42
TSHR P16473 1/20 0.42
ABCB1 P08183 1/20 0.39
ADORA3 P0DMS8 2/20 0.39
MAPT P10636 1/20 0.39
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
IDO1 P14902 1/20 0.39
PDE5A O76074 1/20 0.38
PDE4A P27815 1/20 0.38
PDE1A P54750 1/20 0.38
PDE1B Q01064 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10692521 0.81 KDM4E (0.40) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL7771748 0.76 HSD17B1 (0.46) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL1355596 0.76 ALDH1A1 (0.45) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL6774791 0.74 BRD4 (0.55) ALDH1A1KMT2AMEN1TSHRADORA3
SCHEMBL76231 0.72 ACHE (0.48) ALDH1A1KMT2AMEN1MAPTKDM4E
SCHEMBL7140477 0.72 TUBB4A (0.46) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL11456734 0.71 KDM4E (0.49) ALDH1A1KMT2ATSHRMAPTKDM4E
SCHEMBL7959158 0.71 PDE5A (0.45) ALDH1A1KMT2AMEN1TSHRABCB1
SCHEMBL26850914 0.71 ABCB1 (0.47) ALDH1A1KMT2AMEN1TSHRABCB1
SCHEMBL8531955 0.71 MEN1 (0.48) ALDH1A1KMT2AMEN1TSHRABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673092-B1 HETEROCYCLE-SUBSTITUTED PTERIDINE DERIVATIVES AND THEIR USE IN THERAPY 4 AZA IP NV (BE) 2007-08-15 EP disclosed
EP-1673092-A1 HETEROCYCLE-SUBSTITUTED PTERIDINE DERIVATIVES AND THEIR USE IN THERAPY 4 AZA Bioscience nv (BE) 2006-06-28 EP disclosed
WO-2005039587-A1 HETEROCYCLE-SUBSTITUTED PTERIDINE DERIVATIVES AND THEIR USE IN THERAPY 4 AZA BIOSCIENCE NV (BE) 2005-05-06 WO disclosed