SCHEMBL10692536

SCHEMBL10692536

CN1C(=O)C(C)(c2ccccc2O)Cc2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
POLB P06746 1/20 0.40
MAPT P10636 4/20 0.39
KDM4E B2RXH2 2/20 0.39
LMNA P02545 2/20 0.39
HCRTR1 O43613 1/20 0.39
NPC1 O15118 1/20 0.39
EHMT2 Q96KQ7 1/20 0.39
RAD52 P43351 1/20 0.39
MAPK1 P28482 1/20 0.38
ADAMTS5 Q9UNA0 2/20 0.38
ALDH1A1 P00352 1/20 0.37
PKM P14618 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
BACE1 P56817 3/20 0.36
NQO1 P15559 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10689170 0.81 ADRA1A (0.40) TSHRHTTMAPTKDM4EMAPK1
SCHEMBL10694392 0.80 NPC1 (0.47) NOTUMTSHRHTTPOLBMAPT
SCHEMBL10695401 0.80 RAD52 (0.42) NOTUMTSHRHTTMAPTKDM4E
SCHEMBL10692682 0.77 NPC1 (0.47) HTTMAPTKDM4ELMNAHCRTR1
SCHEMBL2470209 0.75 NOTUM (0.46) NOTUMTSHRHTTMAPTKDM4E
SCHEMBL10694080 0.74 NPC1 (0.45) NPC1EHMT2
SCHEMBL15314930 0.71 RAB9A (0.53) TSHRHTTMAPTKDM4ELMNA
SCHEMBL9590671 0.69 NOTUM (0.44) NOTUMTSHRHTTMAPTKDM4E
SCHEMBL27019600 0.69 EHMT2 (0.44) NOTUMTSHRHTTMAPTKDM4E
SCHEMBL10371341 0.68 RAD52 (0.54) TSHRMAPTKDM4ELMNAHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed