SCHEMBL10694080

SCHEMBL10694080

CCCCCCC1(c2ccccc2O)Cc2ccccc2N(C)C1=O

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
HTR7 P34969 5/20 0.40
OPRL1 P41146 1/20 0.39
HTR1A P08908 1/20 0.39
SIGMAR1 Q99720 4/20 0.38
SCN9A Q15858 5/20 0.37
SLC6A2 P23975 2/20 0.36
EHMT2 Q96KQ7 1/20 0.35
IDH1 O75874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694392 0.86 NPC1 (0.47) NPC1HTR7OPRL1EHMT2
SCHEMBL10691444 0.84 ALDH1A1 (0.43) HTR7OPRL1HTR1ASCN9A
SCHEMBL10692682 0.80 NPC1 (0.47) NPC1EHMT2
SCHEMBL10692777 0.79 OPRL1 (0.35) HTR7OPRL1HTR1ASCN9A
SCHEMBL10692536 0.74 NOTUM (0.41) NPC1EHMT2
SCHEMBL10695401 0.71 RAD52 (0.42) NPC1OPRL1EHMT2
SCHEMBL10690604 0.69 TDP1 (0.42) HTR7SCN9A
SCHEMBL10780105 0.67 CNR1 (0.49) OPRL1SIGMAR1
SCHEMBL27019600 0.67 EHMT2 (0.44) SLC6A2EHMT2
SCHEMBL10694109 0.66 POLB (0.35) HTR7SLC6A2EHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed