SCHEMBL10693440

SCHEMBL10693440

Cc1nnc2n1-c1ccc(OCCN3CCOCC3)cc1C(c1ccccc1Cl)=NC2

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.60
GABRA5 P31644 4/20 0.60
GABRA2 P47869 4/20 0.60
GABRA3 P34903 3/20 0.60
OPRK1 P41145 2/20 0.60
PDE4D Q08499 2/20 0.60
GABRG2 P18507 1/20 0.60
HTR2A P28223 1/20 0.60
GABRB3 P28472 1/20 0.60
ADRA1A P35348 1/20 0.60
GABRB2 P47870 3/20 0.59
PTAFR P25105 9/20 0.58
TSHR P16473 1/20 0.58
ALDH1A1 P00352 2/20 0.54
MEN1 O00255 1/20 0.54
LMNA P02545 1/20 0.54
GAA P10253 1/20 0.54
MAPT P10636 1/20 0.54
HTT P42858 1/20 0.54
KMT2A Q03164 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694618 0.89 GABRA1 (0.56) GABRA1GABRA5GABRA2GABRA3OPRK1
SCHEMBL10698677 0.84 GABRA1 (0.56) GABRA1GABRA5GABRA2GABRA3OPRK1
SCHEMBL10691840 0.83 PTAFR (0.68) GABRA1GABRA5GABRA2GABRA3OPRK1
SCHEMBL11681893 0.78 GABRA1 (0.69) GABRA1GABRA5GABRA2GABRA3OPRK1
SCHEMBL10692488 0.78 GABRA1 (0.62) GABRA1GABRA5GABRA2GABRA3OPRK1
SCHEMBL9668954 0.77 PTAFR (0.74) OPRK1PDE4DPTAFRCYP3A4ALOX15
Triazolam SCHEMBL29228 0.76 GABRA1 (1.00) GABRA1GABRA5GABRA2GABRA3OPRK1
SCHEMBL13352295 0.76 GABRA1 (0.83) GABRA1GABRA5GABRA2GABRA3OPRK1
Triazolam SCHEMBL5142333 0.76 GABRA1 (1.00) GABRA1GABRA5GABRA2GABRA3OPRK1
SCHEMBL10694341 0.76 NPC1 (0.48) PTAFRTSHRALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0255028-A2 1,4-Benzodiazepines, their preparation and use as PAF antagonists BOEHRINGER INGELHEIM KG (DE) 1988-02-03 EP disclosed