SCHEMBL10694341

SCHEMBL10694341

Cc1nnc2n1-c1ccc(OCCN3CCOCC3)cc1C(c1ccccc1Cl)NC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.48
PTAFR P25105 2/20 0.47
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 1/20 0.46
PDE2A O00408 1/20 0.45
OXTR P30559 1/20 0.43
AVPR1A P37288 1/20 0.43
BRD4 O60885 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
MET P08581 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAOA P21397 1/20 0.40
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
RAB9A P51151 1/20 0.39
FGFR1 P11362 1/20 0.39
SRC P12931 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694493 0.79 PTAFR (0.47) PTAFRKDM4EALDH1A1MEN1KMT2A
SCHEMBL10693440 0.76 GABRA1 (0.60) NPC1PTAFRALDH1A1PDE2AMEN1
SCHEMBL10470823 0.75 PTAFR (0.44) PTAFR
SCHEMBL10694618 0.71 GABRA1 (0.56) NPC1PDE2AOXTRAVPR1ABRD4
SCHEMBL9653808 0.69 PTAFR (0.48) PTAFRBRD4
Hydrochloric Acid SCHEMBL9651260 0.68 PTAFR (0.47) PTAFRBRD4
SCHEMBL10698677 0.67 GABRA1 (0.56) OXTRAVPR1ABRD4FGFR1SRC
SCHEMBL11541215 0.67 NPC1 (0.51) NPC1KDM4EALDH1A1METMEN1
SCHEMBL259795 0.64 NPC1 (0.77) NPC1KDM4EALDH1A1SIGMAR1MEN1
SCHEMBL4420934 0.64 NPC1 (0.65) NPC1KDM4EALDH1A1SIGMAR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0255028-A2 1,4-Benzodiazepines, their preparation and use as PAF antagonists BOEHRINGER INGELHEIM KG (DE) 1988-02-03 EP disclosed