SCHEMBL10694618

SCHEMBL10694618

Cc1nnc2n1-c1ccc(OCCN3CCOCC3)cc1C(c1ccccc1)=NC2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 7/20 0.56
GABRA5 P31644 7/20 0.56
GABRA2 P47869 7/20 0.56
GABRB2 P47870 6/20 0.56
GABRA3 P34903 5/20 0.56
HPGD P15428 3/20 0.56
OPRK1 P41145 3/20 0.56
BRD4 O60885 2/20 0.56
LMNA P02545 1/20 0.56
CNR1 P21554 1/20 0.56
OXTR P30559 1/20 0.52
AVPR1A P37288 1/20 0.52
NPC1 O15118 2/20 0.48
RAB9A P51151 1/20 0.48
PPARG P37231 3/20 0.48
ADORA3 P0DMS8 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA2B P29275 1/20 0.45
ADORA1 P30542 1/20 0.45
PDE2A O00408 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698677 0.96 GABRA1 (0.56) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL10693440 0.89 GABRA1 (0.60) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL10694413 0.83 MAPK1 (0.45) LMNANPC1RAB9APPARGADORA3
SCHEMBL7318994 0.80 GABRA1 (0.71) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL10694270 0.79 GABRA1 (0.62) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL10694252 0.76 GABRA1 (0.58) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL8250450 0.73 GABRA1 (0.74) GABRA1GABRA5GABRA2GABRB2GABRA3
Alprazolam SCHEMBL5480614 0.73 GABRA1 (1.00) GABRA1GABRA5GABRA2GABRB2GABRA3
Alprazolam SCHEMBL16922178 0.73 GABRA1 (1.00) GABRA1GABRA5GABRA2GABRB2GABRA3
Alprazolam SCHEMBL8398 0.73 GABRA1 (1.00) GABRA1GABRA5GABRA2GABRB2GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0255028-A2 1,4-Benzodiazepines, their preparation and use as PAF antagonists BOEHRINGER INGELHEIM KG (DE) 1988-02-03 EP disclosed