SCHEMBL10692777

SCHEMBL10692777

CCCCCCC1(c2ccccc2OCCCCBr)Cc2ccccc2N(C)C1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 1/20 0.35
HTR7 P34969 5/20 0.34
S1PR5 Q9H228 1/20 0.34
PRKCA P17252 1/20 0.34
MEN1 O00255 1/20 0.34
NR1I2 O75469 1/20 0.34
LMNA P02545 1/20 0.34
CHRM2 P08172 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADRA2A P08913 1/20 0.34
MAPT P10636 1/20 0.34
OPRK1 P41145 1/20 0.34
HTR2B P41595 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KMT2A Q03164 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SCN9A Q15858 3/20 0.33
HTR1A P08908 1/20 0.33
NAMPT P43490 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694109 0.89 POLB (0.35) HTR7LMNAMAPTALDH1A1DRD2
SCHEMBL10691444 0.86 ALDH1A1 (0.43) OPRL1HTR7ALDH1A1SCN9AHTR1A
SCHEMBL10694576 0.84 POLB (0.33) HTR7LMNAMAPTALDH1A1DRD2
SCHEMBL10690584 0.81 ALDH1A1 (0.36) OPRL1MAPTOPRK1ALDH1A1HTR1A
SCHEMBL10755079 0.80 HTR1A (0.40) OPRL1HTR7ALDH1A1HTR1ADRD2
SCHEMBL10694080 0.79 NPC1 (0.45) OPRL1HTR7SCN9AHTR1A
SCHEMBL10696619 0.79 RAD52 (0.34) OPRL1MAPTOPRK1ALDH1A1HTR1A
SCHEMBL10693548 0.78 RAD52 (0.35) OPRL1MAPTOPRK1ALDH1A1HTR1A
Oxalic Acid SCHEMBL10688530 0.77 SMPD1 (0.45) MAPTALDH1A1
Hydrochloric Acid SCHEMBL10688129 0.77 ALDH1A1 (0.38) OPRL1HTR7ALDH1A1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed