SCHEMBL10695586

SCHEMBL10695586

N#Cc1[nH]c(-c2ccccc2C(F)(F)F)nc1C(N)=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.57
HDAC3 O15379 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
SCN9A Q15858 3/20 0.42
TRPA1 O75762 1/20 0.39
CTSK P43235 1/20 0.39
PDE10A Q9Y233 1/20 0.38
AR P10275 1/20 0.37
KMO O15229 1/20 0.37
CDC7 O00311 1/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
DBF4 Q9UBU7 1/20 0.36
SLC9A1 P19634 1/20 0.36
ATR Q13535 1/20 0.36
FFAR1 O14842 1/20 0.36
LGMN Q99538 1/20 0.36
PIP4K2A P48426 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694425 0.83 PARP1 (0.54) PARP1CDC7SLC9A1
SCHEMBL10694398 0.81 SLC9A1 (0.54) PARP1SLC9A1
SCHEMBL10695611 0.81 PARP1 (0.54) PARP1SLC9A1
SCHEMBL10695343 0.79 PARP1 (0.45) PARP1HDAC3HDAC7HDAC10HDAC6
SCHEMBL10694101 0.77 PARP1 (0.54) PARP1
Valine SCHEMBL10695541 0.73 SLC9A1 (0.45) PARP1SLC9A1LGMN
SCHEMBL7320347 0.72 PARP1 (1.00) PARP1
SCHEMBL10695803 0.72 CHEK2 (0.47) PARP1HDAC3HDAC6
SCHEMBL9220531 0.72 NPBWR1 (0.36) PARP1
SCHEMBL10694053 0.72 CHEK2 (0.48) PARP1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269238-A1 Imidazoles and their compositions for plant growth regulation MAY & BAKER LIMITED (GB) 1988-06-01 EP disclosed