SCHEMBL10696420

SCHEMBL10696420

CC1(C)C(=O)N(Cc2ccccc2)c2cc3c(cc21)NC(c1cccnc1)N3

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.43
ALDH1A1 P00352 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
TP53 P04637 1/20 0.40
MDM2 Q00987 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
RECQL P46063 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
MCL1 Q07820 1/20 0.39
TSHR P16473 1/20 0.38
HDAC1 Q13547 3/20 0.37
HDAC6 Q9UBN7 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694215 0.89 ELANE (0.46) ELANEALDH1A1TP53TDP1KDM4E
SCHEMBL10700217 0.87 KDM4E (0.41) ALDH1A1CYP3A4CYP2C19KDM4EMEN1
SCHEMBL10696318 0.86 KDM4E (0.41) ALDH1A1SMN1; SMN2CYP3A4CYP2C19KDM4E
SCHEMBL10697577 0.85 KDM4E (0.40) ALDH1A1SMN1; SMN2CYP3A4CYP2C9CYP2C19
SCHEMBL10696477 0.84 KDM4E (0.42) ALDH1A1SMN1; SMN2CYP3A4CYP2C9CYP2C19
SCHEMBL10698284 0.84 MEN1 (0.39) ALDH1A1SMN1; SMN2CYP3A4CYP2C9TDP1
SCHEMBL10695491 0.84 MAPT (0.42) ALDH1A1SMN1; SMN2CYP3A4CYP2C19KDM4E
SCHEMBL10691679 0.82 KDM4E (0.45) ALDH1A1CYP3A4CYP2C19KDM4EMEN1
SCHEMBL10696048 0.82 ELANE (0.44) ELANEALDH1A1SMN1; SMN2CYP3A4CYP2C9
SCHEMBL10696091 0.80 TDP1 (0.54) ELANEALDH1A1CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed