SCHEMBL10700809

SCHEMBL10700809

CCN1C(=O)C(C)(C)c2cc3c(cc21)NC(c1ccc([N+](=O)[O-])cc1)N3

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
GAA P10253 4/20 0.43
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
MAPT P10636 2/20 0.43
GFER P55789 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
KDM4E B2RXH2 3/20 0.36
HSPA9 P38646 2/20 0.36
POLB P06746 2/20 0.36
LMNA P02545 1/20 0.35
RECQL P46063 1/20 0.35
CYP1A2 P05177 1/20 0.34
AKR1B1 P15121 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698153 0.85 AURKA (0.38) AURKAAURKBHSPA9
SCHEMBL10698519 0.85 CNR1 (0.41) ALDH1A1GAAKMT2AMEN1AURKA
SCHEMBL10696324 0.84 AURKA (0.36) AURKAAURKB
SCHEMBL10699847 0.84 AURKA (0.39) GAAKMT2AMEN1MAPTAURKA
SCHEMBL10701198 0.83 TNKS2 (0.44) ALDH1A1GAAKMT2AMEN1MAPT
SCHEMBL10699045 0.83 GAA (0.42) ALDH1A1GAAKMT2AMEN1MAPT
SCHEMBL10697456 0.83 MEN1 (0.40) ALDH1A1GAAKMT2AMEN1MAPT
SCHEMBL10699585 0.83 PGR (0.39) AURKAAURKB
SCHEMBL10696613 0.82 AURKA (0.40) ALDH1A1GAAKMT2AAURKAAURKB
SCHEMBL10705923 0.79 GAA (0.42) ALDH1A1GAAKMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed