SCHEMBL10696324

SCHEMBL10696324

CCN1C(=O)C(C)(C)c2cc3c(cc21)NC(c1ccc([S+](C)[O-])cc1)N3

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.36
AURKB Q96GD4 2/20 0.36
CHEK1 O14757 1/20 0.35
SRC P12931 1/20 0.35
CDK2 P24941 1/20 0.35
KDR P35968 1/20 0.35
FLT3 P36888 1/20 0.35
GSK3B P49841 1/20 0.35
BRD4 O60885 1/20 0.32
PGR P06401 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698153 0.85 AURKA (0.38) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10698519 0.85 CNR1 (0.41) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10700809 0.84 ALDH1A1 (0.43) AURKAAURKB
SCHEMBL10699847 0.84 AURKA (0.39) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10699585 0.83 PGR (0.39) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10697456 0.83 MEN1 (0.40) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10699045 0.83 GAA (0.42) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10701198 0.83 TNKS2 (0.44) AURKAAURKBPGR
SCHEMBL10696613 0.82 AURKA (0.40) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10705923 0.79 GAA (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed