SCHEMBL10698519

SCHEMBL10698519

CCN1C(=O)C(C)(C)c2cc3c(cc21)NC(c1ccc(O)cc1)N3

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.41
GPR55 Q9Y2T6 2/20 0.41
KMT2A Q03164 3/20 0.40
AURKA O14965 2/20 0.38
AURKB Q96GD4 2/20 0.38
MEN1 O00255 2/20 0.36
GAA P10253 1/20 0.36
AR P10275 1/20 0.36
IDE P14735 1/20 0.36
ALDH1A1 P00352 3/20 0.35
HTT P42858 2/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
CHEK1 O14757 1/20 0.35
SRC P12931 1/20 0.35
CDK2 P24941 1/20 0.35
KDR P35968 1/20 0.35
FLT3 P36888 1/20 0.35
GSK3B P49841 1/20 0.35
ESR1 P03372 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698153 0.88 AURKA (0.38) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10698974 0.86 KMT2A (0.37) KMT2AMEN1GAAARIDE
SCHEMBL10699585 0.86 PGR (0.39) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10697456 0.86 MEN1 (0.40) CNR1GPR55KMT2AAURKAAURKB
SCHEMBL10699045 0.86 GAA (0.42) KMT2AAURKAAURKBMEN1GAA
SCHEMBL10701198 0.86 TNKS2 (0.44) KMT2AAURKAAURKBMEN1GAA
SCHEMBL10696613 0.85 AURKA (0.40) KMT2AAURKAAURKBGAAAR
SCHEMBL10696324 0.85 AURKA (0.36) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10700809 0.85 ALDH1A1 (0.43) KMT2AAURKAAURKBMEN1GAA
SCHEMBL10705923 0.84 GAA (0.42) KMT2AMEN1GAAALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed