SCHEMBL10698153

SCHEMBL10698153

CCN1C(=O)C(C)(C)c2cc3c(cc21)NC(c1ccc(N)cc1)N3

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.38
AURKB Q96GD4 2/20 0.38
CYP19A1 P11511 12/20 0.36
CHEK1 O14757 1/20 0.35
SRC P12931 1/20 0.35
CDK2 P24941 1/20 0.35
KDR P35968 1/20 0.35
FLT3 P36888 1/20 0.35
GSK3B P49841 1/20 0.35
BRD4 O60885 1/20 0.33
ATAD2 Q6PL18 1/20 0.33
HSPA9 P38646 1/20 0.32
PGR P06401 1/20 0.32
MARK3 P27448 1/20 0.31
ALPL P05186 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698519 0.88 CNR1 (0.41) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10697456 0.86 MEN1 (0.40) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10699585 0.86 PGR (0.39) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10701198 0.86 TNKS2 (0.44) AURKAAURKBPGR
SCHEMBL10699045 0.86 GAA (0.42) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10696613 0.85 AURKA (0.40) AURKAAURKBCYP19A1CHEK1SRC
SCHEMBL10696324 0.85 AURKA (0.36) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10700809 0.85 ALDH1A1 (0.43) AURKAAURKBHSPA9
SCHEMBL10698038 0.84 AURKA (0.40) AURKAAURKBCHEK1SRCCDK2
SCHEMBL10697557 0.83 AURKA (0.37) AURKAAURKBCHEK1SRCCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed