SCHEMBL10706018

SCHEMBL10706018

O=C(N[C@@H](Cc1ccccc1)C(=O)NC1CCCCC1)OCc1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSL P07711 5/20 0.64
ALDH1A1 P00352 2/20 0.64
EPHX1 P07099 1/20 0.62
TACR1 P25103 2/20 0.60
CTSK P43235 6/20 0.59
KDM4E B2RXH2 1/20 0.59
CTSS P25774 4/20 0.59
CTSB P07858 3/20 0.59
HDAC1 Q13547 1/20 0.58
HDAC2 Q92769 1/20 0.58
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8817011 0.94 EPHX1 (0.58) CTSLALDH1A1EPHX1TACR1CTSK
SCHEMBL8817014 0.94 EPHX1 (0.58) CTSLALDH1A1EPHX1TACR1CTSK
SCHEMBL26477860 0.86 EPHX1 (0.57) CTSLALDH1A1EPHX1CTSKCTSS
SCHEMBL11431644 0.84 ALDH1A1 (0.61) ALDH1A1EPHX1CTSKHDAC1HDAC2
Bicarbonate SCHEMBL3824417 0.84 HDAC1 (0.55) CTSLALDH1A1EPHX1CTSKCTSS
SCHEMBL12856074 0.84 L3MBTL1 (0.60) CTSLALDH1A1EPHX1KDM4EHDAC1
SCHEMBL11024260 0.84 TACR1 (0.58) CTSLTACR1CTSKCTSSCTSB
SCHEMBL26477889 0.83 HDAC1 (0.64) ALDH1A1EPHX1CTSKHDAC1HDAC2
SCHEMBL7855475 0.83 ACE (0.54) CTSLALDH1A1EPHX1CTSKKDM4E
Hydrochloric Acid SCHEMBL7851195 0.82 ACE (0.53) CTSLALDH1A1EPHX1CTSKKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0135183-B1 PROCESS FOR THE PREPARATION OF COMPOUNDS CONTAINING CARBOXYLIC ACID AMIDE GROUPS, ESPECIALLY OF PEPTIDES HOECHST AKTIENGESELLSCHAFT (DE) 1988-03-30 EP disclosed
EP-0135183-A2 Process for the preparation of compounds containing carboxylic acid amide groups, especially of peptides HOECHST AKTIENGESELLSCHAFT (DE) 1985-03-27 EP disclosed