SCHEMBL8559411

SCHEMBL8559411

Oc1ccc2[nH]cc(C3CCN(CCCc4c[nH]c5ccccc45)CC3)c2c1

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.61
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
THPO P40225 1/20 0.60
ADRA1D P25100 4/20 0.59
SLC6A4 P31645 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556970 0.97 ADRA1D (0.60) HTR1ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8554847 0.94 CYP1A2 (0.65) HTR1ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8558927 0.93 ADRA1D (0.63) HTR1ACYP1A2CYP3A4CYP2C9ADRA1D
SCHEMBL8559641 0.90 CYP1A2 (0.63) HTR1ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8559023 0.90 CYP1A2 (0.60) HTR1ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8554922 0.89 ADRA1D (0.73) HTR1AADRA1DSLC6A4
SCHEMBL7533736 0.87 CYP1A2 (0.62) CYP1A2CYP3A4CYP2D6CYP2C9THPO
SCHEMBL8556391 0.86 ADRA1D (0.74) HTR1AADRA1DSLC6A4
SCHEMBL8558241 0.85 HTR1A (0.69) HTR1ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8558005 0.85 HTR1A (0.77) HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683166-B1 3-Indolylpiperidines MERCK PATENT GMBH (DE) 1998-10-28 EP disclosed
EP-0683166-A1 3-Indolylpiperidines MERCK PATENT GmbH (DE) 1995-11-22 EP disclosed