SCHEMBL1075112

SCHEMBL1075112

O=C1Nc2ccc(Oc3cccc4c3C(=O)C(=O)N4)cc2C1=O

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 6/20 0.67
MAOB P27338 11/20 0.62
MAOA P21397 10/20 0.62
ALDH1A1 P00352 1/20 0.55
CES1 P23141 5/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1027756 0.81 TGM2 (1.00) TGM2MAOBMAOAALDH1A1CES1
5-Methoxyisatin SCHEMBL28560213 0.72 ALDH1A1 (0.84) TGM2MAOBMAOAALDH1A1CES1
5-Methoxyisatin SCHEMBL29506298 0.72 ALDH1A1 (1.00) TGM2MAOBMAOAALDH1A1CES1
5-Methoxyisatin SCHEMBL21602 0.72 ALDH1A1 (1.00) TGM2MAOBMAOAALDH1A1CES1
SCHEMBL281586 0.72 CES1 (0.55) TGM2MAOBMAOAALDH1A1CES1
SCHEMBL30397534 0.72 CES1 (0.55) TGM2MAOBMAOAALDH1A1CES1
5-Methoxyisatin SCHEMBL3935863 0.70 ALDH1A1 (0.96) TGM2MAOBMAOAALDH1A1CES1
SCHEMBL28812042 0.69 MAOA (0.59) MAOBMAOA
SCHEMBL23385135 0.69 TGM2 (0.71) TGM2MAOBMAOAALDH1A1CES1
Isatin SCHEMBL28259465 0.69 CES1 (0.86) TGM2MAOBMAOAALDH1A1CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274280-A2 BIS-ARYL COMPOUNDS FOR USE AS MEDICAMENTS Biolipox AB (SE) 2011-01-19 EP disclosed
WO-2009127822-A2 BIS-ARYL COMPOUNDS FOR USE AS MEDICAMENTS BIOLIPOX AB (SE) 2009-10-22 WO disclosed