5-Methoxyisatin

5-Methoxyisatin

SCHEMBL21602

COc1ccc2c(c1)C(=O)C(=O)N2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 1.00
TGM2 P21980 6/20 0.73
MAOB P27338 5/20 0.63
MAOA P21397 4/20 0.63
CES1 P23141 4/20 0.63
LRRK2 Q5S007 2/20 0.58
PDE3B Q13370 1/20 0.58
PDE3A Q14432 1/20 0.58
MAPT P10636 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
TLK2 Q86UE8 2/20 0.54
PDPK1 O15530 1/20 0.54
RET P07949 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
5-Methoxyisatin SCHEMBL29506298 1.00 ALDH1A1 (1.00) ALDH1A1TGM2MAOBMAOACES1
5-Methoxyisatin SCHEMBL3935863 0.98 ALDH1A1 (0.96) ALDH1A1TGM2MAOBMAOACES1
5-Methoxyisatin SCHEMBL28560213 0.92 ALDH1A1 (0.84) ALDH1A1TGM2MAOBMAOACES1
SCHEMBL1249793 0.85 ALDH1A1 (0.74) ALDH1A1TGM2MAOBMAOACES1
SCHEMBL1027756 0.85 TGM2 (1.00) ALDH1A1TGM2MAOBMAOACES1
SCHEMBL21179898 0.82 ALDH1A1 (0.70) ALDH1A1TGM2LRRK2PDE3BPDE3A
SCHEMBL2372943 0.81 ALDH1A1 (0.68) ALDH1A1TGM2MAOBMAOACES1
SCHEMBL5918370 0.81 ALDH1A1 (0.68) ALDH1A1LRRK2PDE3BPDE3AMAPT
SCHEMBL19928099 0.80 ALDH1A1 (0.66) ALDH1A1LRRK2PDE3BPDE3AMAPT
SCHEMBL20246772 0.80 ALDH1A1 (0.66) ALDH1A1LRRK2PDE3BPDE3AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 938 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119707805-A Preparation method of 6-hydroxyquinoline-4-carboxylic acid 上海德浦生物医药科技有限公司 2025-03-28 CN claimed
CN-119350241-A Quinolinone derivative and preparation method and application thereof 浙江工业大学 2025-01-24 CN claimed
CN-118852031-A 2, 3-Disubstituted quinazolinone compound and preparation method thereof 赣南师范大学 2024-10-29 CN claimed
CN-113912609-B Preparation method of natural alkaloid tryptanthrin and derivatives thereof 江苏大学 2024-01-05 CN claimed
US-11708373-B2 5-alkylquinazoline derivative, method of preparing the same, and method of using the same HEFEI UNIVERSITY OF TECHNOLOGY (CN) 2023-07-25 US claimed
CN-111187233-B Polysubstituted benzothiazole and derivative and synthesis method thereof 湘潭大学 2023-05-30 CN claimed
CN-114409684-B Preparation and application of chiral amino zinc alkoxide complex 合肥工业大学 2023-05-26 CN claimed
US-20220185819-A1 5-ALKYLQUINAZOLINE DERIVATIVE, METHOD OF PREPARING THE SAME, AND METHOD OF USING THE SAME HEFEI UNIVERSITY OF TECHNOLOGY (CN) 2022-06-16 US claimed
CN-114409684-A Preparation and application of chiral amino zinc alkoxide complex 合肥工业大学 2022-04-29 CN claimed
CN-112480126-B Preparation and application of 5-alkyl quinazoline derivative 合肥工业大学 2022-03-11 CN claimed
EP-1432388-A1 AGENT FOR COLOURING FIBRES CONTAINING KERATIN Henkel Kommanditgesellschaft auf Aktien (DE) 2004-06-30 EP claimed
EP-1432428-A1 Agent for colouring fibres containing keratin Henkel Kommanditgesellschaft auf Aktien (DE) 2004-06-30 EP claimed
EP-1433469-A1 Composition for dyeing keratinous fibres Henkel Kommanditgesellschaft auf Aktien (DE) 2004-06-30 EP claimed
WO-2004022016-A1 AGENTS USED FOR DYEING KERATINOUS FIBERS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2004-03-18 WO claimed
US-6635090-B1 Dyeing method using a specific cationic derivative and a compound selected among a specific aldehyde, a specific ketone, a quinone and a di-imino-isoindoline or 3-amino-isoindolone derivative L'OREAL, S.A. (FR) 2003-10-21 US claimed
WO-2003030847-A1 AGENT FOR COLOURING FIBRES CONTAINING KERATIN HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2003-04-17 WO claimed
WO-2003030842-A1 AGENT FOR COLOURING FIBRES CONTAINING KERATIN HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2003-04-17 WO claimed
EP-1300132-A2 Agent for dyeing keratinous fibres Henkel Kommanditgesellschaft auf Aktien (DE) 2003-04-09 EP claimed
US-6458168-B1 Hair dyeing method using an aliphatic cationic amine and compound chosen from an aldehyde, a ketone, a quinone, a di-imino-isoindoline, and a 3-aminoisoindolone derivative L'OREAL S.A. (FR) 2002-10-01 US claimed
US-6451067-B1 HAIR DYE MIXTURE L'OREAL S.A. (FR) 2002-09-17 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220185819-A1 5-ALKYLQUINAZOLINE DERIVATIVE, METHOD OF PREPARING THE SAME, AND METHOD OF USING THE SAME MLN, PGA5, MCM5 ALDH1A1 4145/4885TGM2 3481/4885MAOB 855/4885
US-11708373-B2 5-alkylquinazoline derivative, method of preparing the same, and method of using the same MLN, MCM5, PGA5 ALDH1A1 3860/4885TGM2 3886/4885MAOB 1449/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.