SCHEMBL1075715

SCHEMBL1075715

Nc1ccc2c(c1)C(O)c1ccccc1-2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 4/20 0.51
HTR7 P34969 2/20 0.51
CDK5 Q00535 1/20 0.47
CDK5R1 Q15078 1/20 0.47
DYRK1A Q13627 1/20 0.47
PDK2 Q15119 3/20 0.46
ALDH1A1 P00352 4/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
LMNA P02545 2/20 0.46
HPGD P15428 2/20 0.46
KDM4E B2RXH2 2/20 0.46
MAPT P10636 2/20 0.46
TP53 P04637 2/20 0.44
CYP3A4 P08684 2/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PTPRC P08575 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL942985 0.89 DYRK1A (0.56) HTR2BHTR7CDK5CDK5R1DYRK1A
SCHEMBL18385982 0.81 HTR2B (0.50) HTR2BHTR7DYRK1AALDH1A1SMN1; SMN2
SCHEMBL29884836 0.80 MAOA (0.52) HTR2BHTR7DYRK1AALDH1A1SMN1; SMN2
SCHEMBL216862 0.80 MAOA (0.52) HTR2BHTR7DYRK1AALDH1A1SMN1; SMN2
SCHEMBL29376368 0.80 MAOA (0.52) HTR2BHTR7DYRK1AALDH1A1SMN1; SMN2
SCHEMBL10632615 0.78 ALDH1A1 (0.56) HTR2BHTR7CDK5CDK5R1ALDH1A1
SCHEMBL27688305 0.78 MAOA (0.50) HTR2BHTR7DYRK1AALDH1A1SMN1; SMN2
SCHEMBL7137182 0.78 HTR7 (0.49) HTR2BHTR7CDK5CDK5R1DYRK1A
SCHEMBL226371 0.78 HTR7 (0.49) HTR2BHTR7CDK5CDK5R1DYRK1A
SCHEMBL5069724 0.78 DYRK1A (0.79) HTR2BHTR7CDK5CDK5R1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 108 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2374853-A1 Cyanate ester-based pressure sensitive adhesive CORNERSTONE RESEARCH GROUP, INC. (US) 2011-10-12 EP claimed
US-20100137554-A1 SHAPE MEMORY CYANATE ESTER COPOLYMERS CORNERSTONE RESEARCH GROUP, INC. 2010-06-03 US claimed
EP-1979397-A4 SHAPE MEMORY CYANATE ESTER COPOLYMERS CORNERSTONE RES GROUP INC (US) 2009-04-08 EP claimed
EP-1979397-A2 SHAPE MEMORY CYANATE ESTER COPOLYMERS CORNERSTONE RESEARCH GROUP, INC. (US) 2008-10-15 EP claimed
WO-2008051241-A2 SHAPE MEMORY CYANATE ESTER COPOLYMERS CORNERSTONE RESEARCH GROUP, INC. (US) 2008-05-02 WO claimed
EP-0667562-B1 Charge injection barrier for positive charging organic photoconductor HEWLETT PACKARD CO (US) 2001-03-21 EP claimed
EP-0515379-A4 ELECTRO-BLOTTING OF ELECTROPHORETICALLY RESOLVED FLUORESCENT-LABELED SACCHARIDES AND DETECTION OF ACTIVE STRUCTURES WITH PROTEIN PROBES GLYCOMED INC (US) 1994-09-14 EP claimed
EP-0515379-A1 ELECTRO-BLOTTING OF ELECTROPHORETICALLY RESOLVED FLUORESCENT-LABELED SACCHARIDES AND DETECTION OF ACTIVE STRUCTURES WITH PROTEIN PROBES GLYCOMED INCORPORATED (US) 1992-12-02 EP claimed
US-5094740-A TWO-DIMENSIONAL ELECTROPHORETIC SEPARATION OF CARBOHYDRATES GLYCOMED, INC. (US) 1992-03-10 US claimed
WO-1991012275-A1 TWO-DIMENSIONAL ELECTROPHORETIC SEPARATION OF CARBOHYDRATES GLYCOMED INCORPORATED (US) 1991-08-22 WO claimed
WO-1991012276-A1 ELECTRO-BLOTTING OF ELECTROPHORETICALLY RESOLVED FLUORESCENT-LABELED SACCHARIDES AND DETECTION OF ACTIVE STRUCTURES WITH PROTEIN PROBES GLYCOMED INCORPORATED (US) 1991-08-22 WO claimed
EP-2277124-B1 MEANS FOR TREATING MYOSIN-RELATED DISEASES HANNOVER MED HOCHSCHULE (DE) 2016-11-09 EP disclosed
US-8536242-B2 Photocurable composition SEKISUI CHEMICAL CO., LTD. (JP) 2013-09-17 US disclosed
EP-1865030-B1 DYE-CONTAINING HARDENABLE COMPOSITION, AND COLOR FILTER AND PROCESS FOR PRODUCING THE SAME FUJIFILM CORP (JP) 2013-06-26 EP disclosed
EP-2175709-B1 SEED TREATMENT METHODS BASF SE (DE) 2013-06-19 EP disclosed
EP-0452696-A2 Aqueous solutions or dispersions of hydroxy-functionalized copolymers, process for their manufacture and use thereof BAYER AG (DE) 1991-10-23 EP disclosed
WO-1991012520-A1 FLUORESCENT TAG FOR SUGAR ELECTROPHORESIS GLYCOMED INCORPORATED (US) 1991-08-22 WO disclosed
WO-1991012276-A1 ELECTRO-BLOTTING OF ELECTROPHORETICALLY RESOLVED FLUORESCENT-LABELED SACCHARIDES AND DETECTION OF ACTIVE STRUCTURES WITH PROTEIN PROBES GLYCOMED INCORPORATED (US) 1991-08-22 WO disclosed
WO-1991012275-A1 TWO-DIMENSIONAL ELECTROPHORETIC SEPARATION OF CARBOHYDRATES GLYCOMED INCORPORATED (US) 1991-08-22 WO disclosed
EP-0401627-A2 Copolymers with hydroxy groups, process for their preparation and their usage as binder BAYER AG (DE) 1990-12-12 EP disclosed