SCHEMBL10848170

SCHEMBL10848170

Nc1cc(N2CCN(Cc3ccccc3)CC2)nc(N2CCN(Cc3ccccc3)CC2)n1

nearest known ligand 0.75

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 8/20 0.75
CASP5 P51878 8/20 0.75
GAA P10253 1/20 0.59
CASP4 P49662 7/20 0.58
HRH4 Q9H3N8 2/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
DRD4 P21917 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
HRH3 Q9Y5N1 1/20 0.49
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
TSHR P16473 1/20 0.48
HTT P42858 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1123752 0.82 CASP1 (0.78) CASP1CASP5GAACASP4NPC1
SCHEMBL10854498 0.81 HRH4 (0.59) CASP1CASP5GAACASP4HRH4
SCHEMBL3991347 0.78 CASP1 (0.67) CASP1CASP5GAACASP4NPC1
SCHEMBL2804769 0.78 CASP1 (0.59) CASP1CASP5GAAHRH4NPC1
SCHEMBL11384876 0.77 CASP1 (0.66) CASP1CASP5GAANPC1RAB9A
SCHEMBL18098559 0.77 CASP1 (0.66) CASP1CASP5GAACASP4NPC1
SCHEMBL477050 0.75 SIGMAR1 (0.55) CASP1CASP5GAANPC1RAB9A
SCHEMBL6685464 0.75 RAB9A (0.59) GAAHRH4NPC1RAB9ALMNA
SCHEMBL3994777 0.75 PIK3CA (0.72) CASP1CASP5
SCHEMBL1083795 0.75 HTR3A (0.68) CASP1CASP5GAAHRH4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4621082-A Pyridopyrimidines, pharmaceutical compositions and use BAYER AKTIENGESELLSCHAFT (DE) 1986-11-04 US disclosed