SCHEMBL1087185

SCHEMBL1087185

CC(C)(C)OC(=O)N[C@@H](Cc1ccc(OC(=O)OC(C)(C)C)cc1)C(=O)O

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.65
ITGA2B P08514 2/20 0.65
ACE P12821 1/20 0.59
PTPN1 P18031 3/20 0.55
CTSS P25774 6/20 0.53
CTSK P43235 5/20 0.53
CTSL P07711 1/20 0.52
CTSB P07858 1/20 0.52
PPARA Q07869 6/20 0.52
PPARG P37231 5/20 0.52
HDAC8 Q9BY41 1/20 0.51
ITGA4 P13612 1/20 0.51
ITGB7 P26010 1/20 0.51
ITGB1 P05556 1/20 0.49
ITGAV P06756 1/20 0.49
ITGB5 P18084 1/20 0.49
PPARD Q03181 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14343235 1.00 ITGB3 (0.65) ITGB3ITGA2BACEPTPN1CTSS
SCHEMBL16909032 1.00 ITGB3 (0.65) ITGB3ITGA2BACEPTPN1CTSS
SCHEMBL8668331 0.90 ITGB3 (0.65) ITGB3ITGA2BACEPTPN1CTSS
SCHEMBL8669351 0.90 ITGB3 (0.65) ITGB3ITGA2BACEPTPN1CTSS
SCHEMBL16993952 0.90 ITGB3 (0.65) ITGB3ITGA2BACEPTPN1CTSS
SCHEMBL5111802 0.89 ITGB3 (0.52) ITGB3ITGA2BACEPTPN1CTSS
SCHEMBL5111794 0.89 ITGB3 (0.52) ITGB3ITGA2BACEPTPN1CTSS
SCHEMBL13654528 0.88 ITGB3 (0.62) ITGB3ITGA2BACEPTPN1CTSS
SCHEMBL3865100 0.87 ITGB3 (0.64) ITGB3ITGA2BACEPTPN1CTSS
SCHEMBL3865096 0.87 ITGB3 (0.64) ITGB3ITGA2BACEPTPN1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12552823-B2 Glucosamine derivatives and pharmaceutical uses thereof Risen (Suzhou) Pharma Tech Co., Ltd. (CN) 2026-02-17 US disclosed
US-20250353870-A1 GLUCOSAMINE DERIVATIVES AND PHARMACEUTICAL USES THEREOF RISEN SUZHOU PHARMA TECH CO LTD (CN) 2025-11-20 US disclosed
US-12312378-B2 Glucosamine derivatives for the prevention or treatment of joint disorders Risen (Suzhou) Pharma Tech Co., Ltd. (CN) 2025-05-27 US disclosed
CN-118290691-A Bio-based antibacterial self-repairing medical polyurethane and preparation method thereof 陕西科技大学 2024-07-05 CN disclosed
US-20240051982-A1 GLUCOSAMINE DERIVATIVES FOR THE PREVENTION OR TREATMENT OF JOINT DISORDERS Risen (Suzhou) Pharma Tech Co., Ltd. (CN) 2024-02-15 US disclosed
US-11718636-B2 Glucosamine derivatives for the prevention or treatment of joint disorders Risen (Suzhou) Pharma Tech Co., Ltd. (CN) 2023-08-08 US disclosed
US-20230227488-A1 GLUCOSAMINE DERIVATIVES AND PHARMACEUTICAL USES THEREOF RISEN SUZHOU PHARMA TECH CO LTD (CN) 2023-07-20 US disclosed
US-11591358-B2 Glucosamine derivatives and pharmaceutical uses thereof Risen (Suzhou) Pharma Tech Co., Ltd. (CN) 2023-02-28 US disclosed
US-20220411461-A1 METHODS OF MAKING INCRETIN ANALOGS ELI LILLY AND COMPANY 2022-12-29 US disclosed
WO-2022185319-A1 UBIQUITIN LIGASE KPC1-PEPTIDE BASED PROTEOLYSIS TARGETING CHIMERAS (PROTAC) AND USES THEREOF TECHNION RESEARCH & DEVELOPMENT FOUNDATION LIMITED (IL) 2022-09-09 WO disclosed
EP-1897550-A2 Prodrugs of Excitatory Amino Acids Eli Lilly & Company (US) 2008-03-12 EP disclosed
US-20060167008-A1 Substituted 1,4,-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists ELANCO ANIMAL HEALTH IRELAND LIMITED (IE) 2006-07-27 US disclosed
US-20050222231-A1 Prodrugs of excitatory amino acids ELI LILLY AND COMPANY (US) 2005-10-06 US disclosed
EP-1551804-A1 SUBSTITUTED 1,4-DI-PIPERIDIN-4-YL-PIPERAZINE DERIVATIVES AND THEIR USE AS NEUROKININ ANTAGONISTS Janssen Pharmaceutica N.V. (BE) 2005-07-13 EP disclosed
WO-2004056772-A1 SUBSTITUTED 1,4-DI-PIPERIDIN-4-YL-PIPERAZINE DERIVATIVES AND THEIR USE AS TACHYKININ ANTAGONISTS JANSSEN PHARMACEUTICA N.V. (BE) 2004-07-08 WO disclosed
WO-2004033428-A1 SUBSTITUTED 1,4-DI-PIPERIDIN-4-YL-PIPERAZINE DERIVATIVES AND THEIR USE AS NEUROKININ ANTAGONISTS JANSSEN PHARMACEUTICA N.V. (BE) 2004-04-22 WO disclosed
EP-0749429-B1 3,5-DISUBSTITUTED AND 3,5,6-TRISUBSTITUTED 2-ISOXAZOLINES AND ISOXAZOLES, PROCESS FOR PREPARING THE SAME AND THEIR USE AS MEDICAMENTS HOECHST AG (DE) 1999-06-30 EP disclosed
US-5814627-A ANTIINFLAMMATORY AGENTS, ASTHMA; RHEUMATIC AND AUTOIMMUNE DISEASES; INHIBITORS OF LEUKOTRIENES, CYTOKINES, E.G. INTERLEUKINS, OXYGEN RADICALS AND PROTEASES HOECHST AKTIENEGESELLSCHAFT (DE) 1998-09-29 US disclosed
EP-0749429-A1 3,5-DISUBSTITUTED AND 3,5,6-TRISUBSTITUTED 2-ISOXAZOLINES AND ISOXAZOLES, PROCESS FOR PREPARING THE SAME AND THEIR USE AS MEDICAMENTS HOECHST AKTIENGESELLSCHAFT (DE) 1996-12-27 EP disclosed
WO-1995024397-A1 3,5-DISUBSTITUTED AND 3,5,6-TRISUBSTITUTED 2-ISOXAZOLINES AND ISOXAZOLES, PROCESS FOR PREPARING THE SAME AND THEIR USE AS MEDICAMENTS HOECHST AKTIENGESELLSCHAFT (DE) 1995-09-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060167008-A1 Substituted 1,4,-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists NPSR1, VIP, TACR1 ITGB3 1543/4885ITGA2B 1388/4885ACE 2095/4885
US-20250353870-A1 GLUCOSAMINE DERIVATIVES AND PHARMACEUTICAL USES THEREOF OGT, UGGT1, GLA ITGB3 1429/4885ITGA2B 1060/4885ACE 605/4885
US-20240051982-A1 GLUCOSAMINE DERIVATIVES FOR THE PREVENTION OR TREATMENT OF JOINT DISORDERS OGT, UGGT1, FUT6 ITGB3 1757/4885ITGA2B 1412/4885ACE 925/4885
US-11718636-B2 Glucosamine derivatives for the prevention or treatment of joint disorders OGT, UGGT1, GLA ITGB3 1927/4885ITGA2B 1511/4885ACE 1293/4885
US-12552823-B2 Glucosamine derivatives and pharmaceutical uses thereof SOST, FUT6, SLC5A1 ITGB3 774/4885ITGA2B 1181/4885ACE 1734/4885
US-20050222231-A1 Prodrugs of excitatory amino acids SLC1A2, SLC1A1, SLC1A3 ITGB3 4476/4885ITGA2B 4089/4885ACE 320/4885
US-20230227488-A1 GLUCOSAMINE DERIVATIVES AND PHARMACEUTICAL USES THEREOF OGT, UGGT1, GLA ITGB3 1429/4885ITGA2B 1060/4885ACE 605/4885
US-20220411461-A1 METHODS OF MAKING INCRETIN ANALOGS IAPP, GLP1R, GIPR ITGB3 4549/4885ITGA2B 4735/4885ACE 736/4885
US-11591358-B2 Glucosamine derivatives and pharmaceutical uses thereof OGT, UGGT1, GLA ITGB3 1429/4885ITGA2B 1060/4885ACE 605/4885
US-12312378-B2 Glucosamine derivatives for the prevention or treatment of joint disorders OGT, UGGT1, FUT6 ITGB3 1757/4885ITGA2B 1412/4885ACE 925/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.