SCHEMBL109244

SCHEMBL109244

C=C(C)C(=O)NCCN(C)CC

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
DNM1 Q05193 1/20 0.33
TGFBR1 P36897 1/20 0.32
NFKB1 P19838 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL111983 0.89 KDM4E (0.41) KDM5AKDM4CKDM4EALDH1A1DNM1
SCHEMBL111490 0.87 KDM5A (0.41) KDM5AKDM4CKDM4EDNM1
SCHEMBL108392 0.86 KDM5A (0.41) KDM5AKDM4CKDM4EDNM1
SCHEMBL522742 0.84 KDM4C (0.41) KDM5AKDM4CKDM4EALDH1A1DNM1
SCHEMBL9414201 0.83 KDM4E (0.35) KDM4ETGFBR1
SCHEMBL93180 0.82 ALDH1A1 (0.47) KDM4EALDH1A1NFKB1KCNH2
SCHEMBL21499 0.82 DNM1 (0.43) KDM4EALDH1A1DNM1
SCHEMBL16271563 0.81 KMT2A (0.37) KDM5AKDM4CTGFBR1
SCHEMBL15270870 0.81 PAOX (0.32) KDM4ETGFBR1
SCHEMBL12655667 0.81 DNM1 (0.45) KDM5AKDM4CDNM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 69 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023107606-A1 BCL-XL/BCL-2 DUAL DEGRADERS FOR TREATMENT OF CANCERS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2023-06-15 WO disclosed
EP-2217827-B1 SUSPENSION SYSTEM FOR AIRCRAFT AUXILIARY POWER UNIT WITH ELASTOMERIC MEMBER LORD CORP (US) 2020-06-03 EP disclosed
EP-3345933-A1 METHOD FOR PRODUCING MODIFIED DIENE RUBBER, RUBBER COMPOSITION, AND TIRE Bridgestone Corporation (JP) 2018-07-11 EP disclosed
EP-2845869-B1 MODIFIED NATURAL RUBBER, METHOD FOR PRODUCING SAME, RUBBER COMPOSITION, AND TIRE BRIDGESTONE CORP (JP) 2018-01-17 EP disclosed
EP-2391339-B1 COLOR-PRESERVING HAIR TREATMENT AGENTS HENKEL AG & CO KGAA (DE) 2017-05-03 EP disclosed
US-9186441-B2 Surface treating agent, filtering material for filter, and blood treatment filter TERUMO KABUSHIKI KAISHA (JP) 2015-11-17 US disclosed
US-9181378-B2 Modified natural rubber and method of manufacturing the same, rubber composition and tire BRIDGESTONE CORPORATION (JP) 2015-11-10 US disclosed
US-9132697-B2 Modified natural rubber or modified natural rubber latex, and rubber composition and pneumatic tire BRIDGESTONE CORPORATION (JP) 2015-09-15 US disclosed
EP-2306967-B1 COLORATION USING CATIONIZABLE POLYMER HENKEL AG & CO KGAA (DE) 2015-07-29 EP disclosed
EP-2845869-A1 MODIFIED NATURAL RUBBER, METHOD FOR PRODUCING SAME, RUBBER COMPOSITION, AND TIRE Bridgestone Corporation (JP) 2015-03-11 EP disclosed
EP-1081162-A1 CONJUGATED DIENE RUBBER, PROCESS FOR PRODUCING THE SAME, AND RUBBER COMPOSITION NIPPON ZEON CO., LTD. (JP) 2001-03-07 EP disclosed
US-6147178-A RUBBER COMPRISING DIENE-VINYL AROMATIC COPOLYMER BEARING QUATERNARY AMMONIUM GROUPS; TENSILE STRENGTH, WEAR RESISTANCE, HEAT RESISTANCE, IMPROVED AFFINITY FOR SILICA REINFORCEMENT NIPPON ZEON CO., LTD. (JP) 2000-11-14 US disclosed
US-6114432-A A DIENE RUBBER COMPONENT INCLUDING AN AMINO GROUP-CONTAINING VINYL MONOMER REINFORCED WITH SILICA; AUTOMOBILE TIRES HAVING EXCELLENT HEAT BUILD-UP RESISTANCE, TENSILE PROPERTIES, ABRASION PROPERTIES AND PROCESSIBILITY NIPPON ZEON CO., LTD. (JP) 2000-09-05 US disclosed
US-6111045-A YIELDS A VULCANIZED RUBBER SHOWING IMPROVEMENTS IN HEAT BUILD-UP, TENSILE STRENGTH, ABRASION RESISTANCE AND PROCESSABILITY NIPPON ZEON CO. LTD. (JP) 2000-08-29 US disclosed
US-6013737-A HAVING IMPROVED TENSILE MODULUS AND IMPROVED ABRASION RESISTANCE, COMPRISING AN AMINO GROUP-CONTAINING DIENE RUBBER OF GIVEN MOONEY VISCOSITY, AND SILICA HAVING SPECIFIC SURFACE AREA, A VULCANIZER AND VULCANIZATION ACCELERATOR NIPPON ZEON CO., LTD. (JP) 2000-01-11 US disclosed
EP-0882738-A1 DIENE RUBBER, PROCESS FOR PRODUCING THE RUBBER AND RUBBER COMPOSITION CONTAINING THE SAME NIPPON ZEON CO., LTD. (JP) 1998-12-09 EP disclosed
EP-0870786-A1 DIENE RUBBER, PROCESS FOR THE PREPARATION OF THE SAME AND COMPOSITION CONTAINING THE SAME NIPPON ZEON CO., LTD. (JP) 1998-10-14 EP disclosed
EP-0864606-A1 RUBBER COMPOSITION NIPPON ZEON CO., LTD. (JP) 1998-09-16 EP disclosed
EP-0849321-A1 DIENE RUBBER COMPOSITION NIPPON ZEON CO., LTD. (JP) 1998-06-24 EP disclosed
EP-0819731-A1 DIENE RUBBER COMPOSITION NIPPON ZEON CO., LTD. (JP) 1998-01-21 EP disclosed