SCHEMBL10936657

SCHEMBL10936657

NCCNc1ccc2cn[nH]c2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
INSR P06213 1/20 0.55
IGF1R P08069 1/20 0.55
ALDH1A1 P00352 9/20 0.54
HSD17B10 Q99714 3/20 0.54
CYP1A2 P05177 2/20 0.54
CYP3A4 P08684 2/20 0.54
CYP2C9 P11712 2/20 0.54
CYP2C19 P33261 2/20 0.54
HIF1A Q16665 2/20 0.54
CYP2D6 P10635 1/20 0.54
PHLPP2 Q6ZVD8 1/20 0.54
MAPT P10636 8/20 0.50
KDM4E B2RXH2 7/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
HTT P42858 2/20 0.50
PIM1 P11309 1/20 0.50
PIM2 Q9P1W9 1/20 0.50
PKM P14618 1/20 0.50
HPGD P15428 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572076 0.87 ROCK2 (0.55) ALDH1A1HIF1AMAPTKDM4EMEN1
SCHEMBL7572085 0.84 RECQL (0.58) INSRIGF1RALDH1A1HSD17B10CYP1A2
SCHEMBL7571372 0.84 INSR (0.58) INSRIGF1RALDH1A1HSD17B10CYP1A2
SCHEMBL7571488 0.80 HPGD (0.62) INSRIGF1RALDH1A1HSD17B10CYP1A2
SCHEMBL13122225 0.78 INSR (0.55) INSRIGF1RALDH1A1HSD17B10CYP1A2
SCHEMBL14911289 0.77 SYK (0.52) HPGDRAB9ANPC1SMN1; SMN2
Hydrochloric Acid SCHEMBL2083483 0.76 ALDH1A1 (0.60) INSRIGF1RALDH1A1HSD17B10CYP1A2
SCHEMBL13122034 0.76 INSR (0.67) INSRIGF1RALDH1A1HSD17B10CYP1A2
SCHEMBL11934937 0.76 ROCK2 (0.51) ALDH1A1HIF1AMAPTKDM4EMEN1
SCHEMBL7572900 0.75 INSR (0.56) INSRIGF1RALDH1A1HSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4507488-A N-Pyrazolylalkylenediamine intermediates BOEHRINGER MANNHEIM GMBH (DE) 1985-03-26 US disclosed
EP-0042592-B1 N-HETEROARYLALKYLENE DIAMINES, PROCESS FOR THEIR PREPARATION AND THEIR USE Roche Diagnostics GmbH (DE) 1985-01-30 EP disclosed