SCHEMBL1095172

SCHEMBL1095172

O=S(=O)(Nc1ccncn1)c1cc(Cl)c(F)cc1F

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 6/20 0.61
SCN8A Q9UQD0 6/20 0.61
SCN1A P35498 5/20 0.61
SCN9A Q15858 15/20 0.58
CYP3A4 P08684 2/20 0.54
CYP2C9 P11712 2/20 0.54
SCN2B O60939 2/20 0.52
SCN1B Q07699 2/20 0.52
SCN2A Q99250 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL20486310 0.99 SCN5A (0.60) SCN5ASCN8ASCN1ASCN9ACYP3A4
SCHEMBL20095679 0.88 SCN5A (0.58) SCN5ASCN8ASCN1ASCN9ACYP3A4
SCHEMBL1093752 0.81 SCN9A (0.58) SCN5ASCN8ASCN1ASCN9A
SCHEMBL17454965 0.81 SCN1A (0.50) SCN5ASCN8ASCN1ASCN9ACYP3A4
SCHEMBL20095711 0.81 SCN9A (0.50) SCN5ASCN8ASCN1ASCN9ACYP3A4
SCHEMBL29835236 0.81 SCN1A (0.59) SCN5ASCN8ASCN1ASCN9ACYP3A4
SCHEMBL23140833 0.80 SCN1A (0.49) SCN5ASCN8ASCN1ASCN9ACYP3A4
SCHEMBL20259316 0.79 SCN1A (0.64) SCN5ASCN8ASCN1ASCN9ASCN1B
SCHEMBL20095732 0.78 SCN1A (0.50) SCN5ASCN8ASCN1ASCN9A
SCHEMBL29482006 0.78 SCN1A (0.50) SCN5ASCN8ASCN1ASCN9ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10316026-B2 Method for removing dimethoxybenzyl group DAIICHI SANKYO COMPANY, LIMITED (JP) 2019-06-11 US disclosed
US-10316026-B2 Method for removing dimethoxybenzyl group DAIICHI SANKYO COMPANY, LIMITED (JP) 2019-06-11 US disclosed
EP-3372583-A1 METHOD FOR REMOVING DIMETHOXYBENZYL GROUP DAIICHI SANKYO COMPANY, LIMITED (JP) 2018-09-12 EP disclosed
US-20180251448-A1 METHOD FOR REMOVING DIMETHOXYBENZYL GROUP DAIICHI SANKYO COMPANY, LIMITED (JP) 2018-09-06 US disclosed
EP-2385938-B1 SULFONAMIDE DERIVATIVES PFIZER LTD (GB) 2015-03-04 EP disclosed
US-8907101-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2014-12-09 US disclosed
US-8907101-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2014-12-09 US disclosed
US-8907101-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2014-12-09 US disclosed
US-20130338111-A1 Sulfonamide Derivatives ICAGEN, INC. (US) 2013-12-19 US disclosed
US-8541588-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2013-09-24 US disclosed
US-20120149679-A1 Sulfonamide Derivatives ICAGEN, INC. 2012-06-14 US disclosed
US-8153814-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2012-04-10 US disclosed
US-8153814-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2012-04-10 US disclosed
US-8153814-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2012-04-10 US disclosed
EP-2385938-A1 SULFONAMIDE DERIVATIVES Pfizer Limited (GB) 2011-11-16 EP disclosed
US-8040476-B2 Display device and method of producing the same MITSUBISHI ELECTRIC CORPORATION (JP) 2011-10-18 US disclosed
US-20100197655-A1 SULFONAMIDE DERIVATIVES Pfizer Limited Icagen, Inc. 2010-08-05 US disclosed
US-20100197655-A1 SULFONAMIDE DERIVATIVES Pfizer Limited Icagen, Inc. 2010-08-05 US disclosed
US-20100197655-A1 SULFONAMIDE DERIVATIVES Pfizer Limited Icagen, Inc. 2010-08-05 US disclosed
WO-2010079443-A1 SULFONAMIDE DERIVATIVES PFIZER LIMITED (GB) 2010-07-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180251448-A1 METHOD FOR REMOVING DIMETHOXYBENZYL GROUP DDT, ALKBH5, DDO SCN5A 4252/4885SCN8A 4661/4885SCN1A 4763/4885
US-20100197655-A1 SULFONAMIDE DERIVATIVES SULT2A1, SULT1A1, TPST2 SCN5A 19/4885SCN8A 32/4885SCN1A 23/4885
US-20130338111-A1 Sulfonamide Derivatives SULT2A1, SULT1A1, TPST2 SCN5A 19/4885SCN8A 32/4885SCN1A 23/4885
US-10316026-B2 Method for removing dimethoxybenzyl group DDT, ALKBH5, DDO SCN5A 4252/4885SCN8A 4661/4885SCN1A 4763/4885
US-20120149679-A1 Sulfonamide Derivatives SULT2A1, SULT1A1, TPST2 SCN5A 19/4885SCN8A 32/4885SCN1A 23/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.