SCHEMBL10957232

SCHEMBL10957232

Cc1cc(CSCCN)oc1CN(C)C

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PRMT6 Q96LA8 1/20 0.59
ACHE P22303 16/20 0.45
BCHE P06276 10/20 0.45
APEX1 P27695 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10959685 0.88 PRMT6 (0.59) PRMT6ACHEBCHE
SCHEMBL11252579 0.84 PRMT6 (0.57) PRMT6ACHEBCHE
SCHEMBL11252584 0.81 PRMT6 (0.55) PRMT6ACHEBCHE
SCHEMBL11254687 0.81 PRMT6 (0.55) PRMT6ACHEBCHEAPEX1
SCHEMBL11253283 0.79 APEX1 (0.52) PRMT6ACHEBCHEAPEX1
SCHEMBL11260097 0.79 PRMT6 (0.52) PRMT6ACHEBCHE
SCHEMBL11244950 0.79 PRMT6 (0.41) PRMT6APEX1
SCHEMBL11460483 0.78 PRMT6 (0.44) PRMT6ACHEBCHE
SCHEMBL10967495 0.77 ACHE (0.36) PRMT6ACHEBCHE
SCHEMBL11479765 0.77 PRMT6 (0.42) PRMT6ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0049049-B1 5-AMINO-TETRAZOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1985-11-13 EP disclosed
US-4536508-A ANTIALLERGENS AND ANTIINFLAMMATORY AGENTS GLAXO GROUP LIMITED (GB) 1985-08-20 US disclosed
US-4510309-A ANTISECRETORY AND ANTIULCER AGENTS BRISTOL-MYERS COMPANY (US) 1985-04-09 US disclosed
US-4471122-A Thiadiazole histamine H2 -antagonists BRISTOL-MYERS COMPANY (US) 1984-09-11 US disclosed
EP-0016565-B1 1,2,4-TRIAZOLE DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1984-05-23 EP disclosed
US-4394508-A ANTIULCER AND ANTISECRETORY AGENTS; HISTAMINE ANTAGONIST BRISTOL-MYERS COMPANY (US) 1983-07-19 US disclosed
US-4380639-A ANTIULCER AND ANTISECRETORY AGENTS BRISTOL-MYERS COMPANY (US) 1983-04-19 US disclosed
US-4380638-A ANTIULCER AND ANTISECRETORY AGENTS; DERIVATIVES OF 3-AMINO-4-HET-A BRISTOL-MYERS COMPANY (US) 1983-04-19 US disclosed
US-4374248-A ANTIHISTAMINES, ANTIULCER BRISTOL-MYERS COMPANY (US) 1983-02-15 US disclosed
EP-0049049-A1 5-Amino-tetrazole derivatives, processes for their preparation and pharmaceutical compositions containing them GLAXO GROUP LIMITED (GB) 1982-04-07 EP disclosed
EP-0001699-B1 DERIVATIVES OF FURYL COMPOUNDS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1982-02-24 EP disclosed
US-4288443-A HISTAMINE ANTAGONISTS GLAXO GROUP LIMITED (GB) 1981-09-08 US disclosed
EP-0016565-A1 1,2,4-Triazole derivatives, processes for their production and pharmaceutical compositions containing them GLAXO GROUP LIMITED (GB) 1980-10-01 EP disclosed
EP-0001699-A2 Derivatives of furyl compounds, their preparation and pharmaceutical compositions containing them GLAXO GROUP LIMITED (GB) 1979-05-02 EP disclosed