SCHEMBL10960645

SCHEMBL10960645

CN(C(=O)OCCCCl)c1cccc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.49
HTR1B P28222 3/20 0.40
LMNA P02545 1/20 0.38
NCEH1 Q6PIU2 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11570035 0.81 SIGMAR1 (0.56) SIGMAR1NCEH1KDM4EALDH1A1HPGD
SCHEMBL6003215 0.80 SIGMAR1 (0.54) SIGMAR1LMNANCEH1ALDH1A1HPGD
SCHEMBL11349063 0.77 CHRNB2 (0.60) LMNACHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL2090835 0.76 SIGMAR1 (0.61) SIGMAR1LMNANCEH1ALDH1A1TSHR
SCHEMBL10963989 0.76 ALDH1A1 (0.40) SIGMAR1HTR1BKDM4EALDH1A1HPGD
SCHEMBL27431595 0.75 SIGMAR1 (0.59) SIGMAR1LMNAKDM4EALDH1A1TSHR
SCHEMBL2090833 0.75 SIGMAR1 (0.59) SIGMAR1LMNANCEH1
SCHEMBL11872011 0.73 SIGMAR1 (0.65) SIGMAR1LMNANCEH1CNR2
SCHEMBL5923592 0.73 SIGMAR1 (0.56) SIGMAR1LMNANCEH1KDM4E
SCHEMBL995336 0.71 CA12 (0.46) SIGMAR1LMNAALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148201-A4 NAPHTALENE AMINOALKYLENE ETHERS AND THIOETHERS, AND THEIR PHARMA CEUTICAL USES. RORER INTERNAT OVERSEAS INC (US) 1985-09-26 EP disclosed
EP-0148201-A1 NAPHTALENE AMINOALKYLENE ETHERS AND THIOETHERS, AND THEIR PHARMA CEUTICAL USES RORER INTERNATIONAL (OVERSEAS) INC. (US) 1985-07-17 EP disclosed
WO-1984004245-A1 NAPHTALENE AMINOALKYLENE ETHERS AND THIOETHERS, AND THEIR PHARMA CEUTICAL USES RORER INT OVERSEAS (US) 1984-11-08 WO disclosed