SCHEMBL1096366

SCHEMBL1096366

C=NNc1ccccc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.48
MEN1 O00255 5/20 0.48
KMT2A Q03164 5/20 0.48
LMNA P02545 3/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
CHRNA7 P36544 1/20 0.41
TSHR P16473 2/20 0.41
HPGD P15428 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CRHBP P24387 1/20 0.40
HTT P42858 1/20 0.40
CRHR2 Q13324 1/20 0.40
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 1/20 0.39
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
APEX1 P27695 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20666032 0.73 TP53 (0.42) MAPTMEN1KMT2ALMNANPC1
SCHEMBL1487981 0.72
SCHEMBL14304537 0.71 GAA (0.46) MAPTMEN1KMT2ALMNANPC1
SCHEMBL20283447 0.71 L3MBTL1 (0.42) MAPTMEN1KMT2ALMNANPC1
SCHEMBL23848857 0.71 POLB (0.43) MAPTMEN1KMT2ARAB9ATSHR
SCHEMBL25078194 0.71 RAB9A (0.45) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL4164253 0.71 MAPT (0.47) MAPTMEN1KMT2ALMNANPC1
SCHEMBL31482338 0.71 LMNA (0.53) MAPTMEN1KMT2ALMNANPC1
SCHEMBL31498989 0.71 TSHR (0.60) MAPTMEN1KMT2ALMNANPC1
SCHEMBL8663534 0.71 LMNA (0.53) MAPTMEN1KMT2ALMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3441390-A1 LIVER X RECEPTOR (LXR) MODULATORS FOR THE TREATMENT OF DERMAL DISEASES, DISORDERS AND CONDITIONS Ralexar Therapeutics, Inc. (US) 2019-02-13 EP disclosed
EP-2820013-B9 LIVER X RECEPTOR (LXR) MODULATORS FOR THE TREATMENT OF DERMAL DISEASES, DISORDERS AND CONDITIONS RALEXAR THERAPEUTICS INC (US) 2019-01-09 EP disclosed
US-8158389-B2 Products and methods for in vivo secretion of monatin CARGILL, INCORPORATED (US) 2012-04-17 US disclosed
US-8153405-B2 Products and methods for in vivo secretion of monatin CARGILL, INCORPORATED (US) 2012-04-10 US disclosed
EP-1883817-A2 PRODUCTS AND METHODS FOR IN VIVO SECRETION OF MONATIN Cargill, Incorporated (US) 2008-02-06 EP disclosed
US-20070105938-A1 Products and Methods for In Vivo Secretion of Monatin CARGILL, INCORPORATED (US) 2007-05-10 US disclosed
US-20070099277-A1 Products and methods for in vivo secretion of monatin CARGILL, INCORPORATED (US) 2007-05-03 US disclosed
WO-2006113897-A2 PRODUCTS AND METHODS FOR IN VIVO SECRETION OF MONATIN CARGILL, INCORPORATED (US) 2006-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070105938-A1 Products and Methods for In Vivo Secretion of Monatin MON2, MLEC, STOM MAPT 4270/4885MEN1 7/4885KMT2A 2730/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.