SCHEMBL10968367

SCHEMBL10968367

O=C(O)C(CCN1C(=O)c2ccccc2C1=O)C(F)F

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 9/20 0.50
MMP9 P14780 9/20 0.50
CA12 O43570 1/20 0.49
CA9 Q16790 1/20 0.49
ALDH1A1 P00352 2/20 0.48
MAPT P10636 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CASP3 P42574 1/20 0.46
HDAC1 Q13547 3/20 0.46
HDAC7 Q8WUI4 3/20 0.46
MMP3 P08254 1/20 0.45
MMP13 P45452 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7080833 0.82 ALDH1A1 (0.58) MMP2MMP9CA12CA9ALDH1A1
SCHEMBL1781793 0.79 ALDH1A1 (0.55) MMP2MMP9CA12CA9ALDH1A1
SCHEMBL1286243 0.79 ALDH1A1 (0.55) MMP2MMP9CA12CA9ALDH1A1
SCHEMBL1841406 0.79 CASP3 (0.55) MMP2MMP9ALDH1A1MAPTSMN1; SMN2
SCHEMBL25234160 0.78 GLS (0.55) ALDH1A1MAPTNPSR1SMN1; SMN2CASP3
SCHEMBL30544887 0.78 GLS (0.55) ALDH1A1MAPTNPSR1SMN1; SMN2CASP3
SCHEMBL7286787 0.78 CA12 (0.51) MMP2MMP9CA12CA9ALDH1A1
SCHEMBL6579299 0.78 MMP2 (0.52) MMP2MMP9CA12CA9ALDH1A1
SCHEMBL7286779 0.78 CA12 (0.51) MMP2MMP9CA12CA9ALDH1A1
SCHEMBL876560 0.78 SMN1; SMN2 (0.53) MMP2MMP9CA12CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0046712-B1 FLUORINATED DIAMINOBUTANE DERIVATIVES MERRELL TORAUDE ET COMPAGNIE (FR) 1985-02-06 EP disclosed
US-4435425-A INHIBITORS OF GAMMA-AMINOBUTYRIC ACID TRANSAMINASE MERRELL TORAUDE ET COMPAGNIE (FR) 1984-03-06 US disclosed
EP-0046712-A1 Fluorinated diaminobutane derivatives MERRELL TORAUDE ET COMPAGNIE (FR) 1982-03-03 EP disclosed