SCHEMBL10977385

SCHEMBL10977385

c1ccc2c(c1)O[C@@H]1CN(CC3CC3)C[C@H]1O2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.47
SIGMAR1 Q99720 2/20 0.38
HTR1A P08908 1/20 0.38
ADRA1D P25100 2/20 0.38
ADRA1A P35348 2/20 0.38
ADRA1B P35368 2/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
SCN1A P35498 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
CHRNB4 P30926 2/20 0.37
CHRNA3 P32297 2/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
CCR1 P32246 3/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10977382 1.00 OPRM1 (0.47) OPRM1SIGMAR1HTR1AADRA1DADRA1A
SCHEMBL10979584 0.77 KMT2A (0.43) ADRA1DADRA1AADRA1BADRA2AADRA2B
SCHEMBL10979581 0.77 KMT2A (0.43) ADRA1DADRA1AADRA1BADRA2AADRA2B
SCHEMBL10977153 0.74 DRD2 (0.42) SIGMAR1CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL10980746 0.74 SIGMAR1 (0.55) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL10977151 0.74 DRD2 (0.42) SIGMAR1CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL10979574 0.74 SIGMAR1 (0.55) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL10980846 0.73 MAOA (0.40) ADRA1DADRA1AADRA1BADRA2AADRA2B
SCHEMBL10980578 0.73 HRH3 (0.49) OPRM1SIGMAR1ADRA1DADRA1AADRA1B
SCHEMBL10980577 0.73 HRH3 (0.49) OPRM1SIGMAR1ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4496579-A AMINATION WITH AMMONIA OR PRIMARY AMINE; ANTIDEPRESANT GLAXO GROUP LIMITED (GB) 1985-01-29 US disclosed