SCHEMBL10992005

SCHEMBL10992005

Cc1cc2ccccc2c(-c2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.48
ADORA1 P30542 2/20 0.48
ALDH1A1 P00352 3/20 0.46
LMNA P02545 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TDO2 P48775 1/20 0.46
MAPK14 Q16539 2/20 0.43
MAPK13 O15264 1/20 0.43
RAF1 P04049 1/20 0.43
MAPK9 P45984 1/20 0.43
MAPK12 P53778 1/20 0.43
MAPK11 Q15759 1/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
ATM Q13315 1/20 0.43
CYP1A2 P05177 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
CYP1A1 P04798 1/20 0.42
CYP1B1 Q16678 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29118704 0.85 DHODH (0.43) NPSR1MAPK14MAPK13RAF1MAPK12
SCHEMBL29118670 0.80 RAB9A (0.43) ADORA1ALDH1A1LMNAMAPK14KMT2A
SCHEMBL25847343 0.80 CYP1A2 (0.42) ADORA2AADORA1ALDH1A1LMNACYP1A2
SCHEMBL10983261 0.79 ADORA2A (0.45) ADORA2AADORA1ALDH1A1LMNANPSR1
SCHEMBL10671008 0.79 PDE10A (0.47) ADORA2AADORA1ALDH1A1LMNAKMT2A
SCHEMBL10986938 0.78 KMO (0.52) ADORA2AADORA1ALDH1A1LMNANPSR1
SCHEMBL11976488 0.78 TDO2 (0.60) ADORA2AADORA1ALDH1A1LMNANPSR1
SCHEMBL8470699 0.77 ABCG2 (0.37) ADORA2AALDH1A1LMNACYP1A2HPGD
SCHEMBL29118727 0.77 NPC1 (0.43) ALDH1A1LMNANPSR1TDO2KMT2A
SCHEMBL10992698 0.77 PARP1 (0.49) ADORA2AADORA1ALDH1A1LMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4499094-A PREVENTION OF RESPIRATORY, UROGENITAL, CARDIOVASCULAR AND IMMUNOLOGICAL DISORDERS WHEN USING FOR BENZDIAPINES PHARMUKA LABORATOIRES (FR) 1985-02-12 US disclosed