SCHEMBL10992502

SCHEMBL10992502

Cn1c(C(=O)CCC(=O)O)cnc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.48
LMNA P02545 2/20 0.45
FFAR1 O14842 1/20 0.45
CYP1A2 P05177 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HIF1A Q16665 1/20 0.45
HPGDS O60760 1/20 0.43
NR4A2 P43354 1/20 0.42
COMT P21964 1/20 0.42
GABRP O00591 3/20 0.40
GABRD O14764 3/20 0.40
GABRA1 P14867 3/20 0.40
GABRB1 P18505 3/20 0.40
GABRG2 P18507 3/20 0.40
GABRB3 P28472 3/20 0.40
GABRA5 P31644 3/20 0.40
GABRA3 P34903 3/20 0.40
GABRA2 P47869 3/20 0.40
GABRB2 P47870 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18356513 0.84 HPGDS (0.44) ESR1LMNARAB9AHPGDSCOMT
SCHEMBL10652832 0.83 HPGDS (0.40) ESR1LMNACYP1A2SMN1; SMN2HIF1A
SCHEMBL2225245 0.81 HPGDS (0.50) ESR1LMNACYP1A2RAB9AHPGDS
SCHEMBL14190000 0.80 HPGDS (0.49) ESR1LMNACYP1A2RAB9ASMN1; SMN2
SCHEMBL4879887 0.78 COMT (0.49) ESR1RAB9ASMN1; SMN2HPGDSCOMT
SCHEMBL6498481 0.77 GABRB2 (0.52) LMNACYP1A2RAB9ASMN1; SMN2GABRA1
SCHEMBL1314013 0.76 RAB9A (0.53) LMNARAB9ASMN1; SMN2HPGDSCOMT
SCHEMBL8669626 0.76 MAP4K4 (0.48) LMNAHPGDSCOMTKMT2APDE3B
SCHEMBL6547472 0.72 CYP11B1 (0.50) ESR1LMNAFFAR1HPGDSCOMT
SCHEMBL10991522 0.71 FFAR1 (0.45) ESR1LMNAFFAR1CYP1A2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521416-A 4,5-Dihydro-6-[(substituted)-1H-imidazol-4-yl or 5-yl]-3(2H)-pyridazinones and 6-[(substituted)-1H-imidazol-4-yl or 5-yl]-3(2H)-pyridazinones WARNER-LAMBERT COMPANY (US) 1985-06-04 US disclosed
EP-0125749-A2 Imidazolyl-pyridazinones WARNER-LAMBERT COMPANY (US) 1984-11-21 EP disclosed