SCHEMBL11000239

SCHEMBL11000239

CCN1C(=O)C=C(c2ccc(Cl)c(Cl)c2)C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RGS4 P49798 1/20 0.44
AHR P35869 3/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
LMNA P02545 3/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
PRKCZ Q05513 1/20 0.36
MAPT P10636 3/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
ALOX12 P18054 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP1B1 Q16678 1/20 0.35
NPSR1 Q6W5P4 2/20 0.34
ALKBH3 Q96Q83 1/20 0.34
CACNA1B Q00975 1/20 0.34
APBA1 Q02410 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11000171 0.79 AHR (0.43) RGS4AHRLMNAKDM4EALDH1A1
SCHEMBL3213620 0.78 GSK3A (0.50) RGS4KDM4EALDH1A1MAPTMEN1
SCHEMBL6809868 0.76 RGS4 (0.48) RGS4LMNAALDH1A1MAPTGAA
SCHEMBL1535501 0.75 RGS4 (0.58) RGS4LMNAALDH1A1MAPTGAA
SCHEMBL3205446 0.74 HTR2A (0.43) RGS4L3MBTL1LMNAKDM4EALDH1A1
SCHEMBL1471569 0.71 RAD51 (0.44) RGS4AHRLMNAALDH1A1MAPT
SCHEMBL20216186 0.69 ALDH1A1 (0.48) RGS4L3MBTL1LMNAKDM4EALDH1A1
SCHEMBL7579280 0.68 MAPT (0.72) RGS4AHRLMNAALDH1A1MAPT
SCHEMBL15355922 0.68 RGS4 (0.41) RGS4LMNAALDH1A1MAPTMEN1
SCHEMBL4774013 0.66 PGR (0.43) LMNAMAPTNPSR1CACNA1BAPBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4529736-A Antidepressant AMERICAN CYANAMID COMPANY (US) 1985-07-16 US disclosed
EP-0100426-A1 3a-(substituted-phenyl)-hexaloctahydro-4,7-alkanoisoindoles AMERICAN CYANAMID COMPANY (US) 1984-02-15 EP disclosed