SCHEMBL11021670

SCHEMBL11021670

CCOc1cc(SC)ccc1-c1nc2cc(C#N)ccc2[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.38
RHEB Q15382 1/20 0.38
S1PR1 P21453 1/20 0.37
METAP2 P50579 1/20 0.36
METAP1 P53582 1/20 0.36
TRPV4 Q9HBA0 1/20 0.36
PKN1 Q16512 1/20 0.36
PKN2 Q16513 1/20 0.36
GUSB P08236 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
RECQL P46063 1/20 0.35
KMT2A Q03164 1/20 0.35
PLG P00747 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11021674 0.92 METAP2 (0.46) PDE5ARHEBMETAP2METAP1PKN1
SCHEMBL10760601 0.88 MAPK10 (0.42) PDE5ARHEBPKN1PKN2MAPK10
SCHEMBL14514686 0.81 RHEB (0.57) PDE5ARHEBS1PR1METAP2METAP1
SCHEMBL10765326 0.81 MAPK10 (0.42) PDE5ARHEBPKN1PKN2MAPK10
SCHEMBL11018065 0.81 PDE5A (0.37) PDE5ARHEBS1PR1METAP2METAP1
SCHEMBL11022213 0.81 ATR (0.44) PDE5ATRPV4GUSBMAPT
SCHEMBL10762222 0.81 AMY1A (0.41) PDE5ARHEBPKN1PKN2KDM4E
Hydrochloric Acid SCHEMBL5647675 0.81 RHEB (0.56) PDE5ARHEBS1PR1METAP2METAP1
SCHEMBL11021081 0.81 CA12 (0.43) PDE5AS1PR1TRPV4GUSBMAPT
SCHEMBL11018823 0.81 TOP1 (0.40) PDE5ARHEBS1PR1METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed