SCHEMBL11021081

SCHEMBL11021081

CCOc1cc(S(N)(=O)=O)ccc1-c1nc2cc(C#N)ccc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.43
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
CA9 Q16790 4/20 0.43
TTK P33981 3/20 0.41
MAPK8 P45983 3/20 0.41
TRPV4 Q9HBA0 1/20 0.41
KMT2A Q03164 1/20 0.40
ATR Q13535 1/20 0.40
PDE5A O76074 1/20 0.38
CA7 P43166 2/20 0.37
CA3 P07451 1/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37
CA5A P35218 1/20 0.37
CA14 Q9ULX7 1/20 0.37
CA5B Q9Y2D0 1/20 0.37
TDP2 O95551 1/20 0.36
GUSB P08236 1/20 0.36
CHEK2 O96017 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11021091 0.92 ATR (0.48) CA12CA1CA2CA9TTK
SCHEMBL11022213 0.91 ATR (0.44) TRPV4ATRPDE5AGUSBBRPF1
SCHEMBL11020313 0.89 CA2 (0.54) CA12CA1CA2CA9ATR
SCHEMBL11021236 0.88 KDM4E (0.42) TRPV4KMT2AATRPDE5ABRPF1
SCHEMBL11021736 0.88 MAPT (0.43) TRPV4KMT2AATRPDE5AGUSB
SCHEMBL11022217 0.83 ATR (0.53) TRPV4ATRCHEK2MAPTSCD
SCHEMBL10763275 0.82 MAPK10 (0.42) CA12CA1CA2CA9PDE5A
SCHEMBL11018065 0.81 PDE5A (0.37) TRPV4KMT2APDE5AGUSBCHEK2
SCHEMBL11020318 0.81 CA12 (0.54) CA12CA1CA2CA9ATR
SCHEMBL11021670 0.81 PDE5A (0.38) TRPV4KMT2APDE5AGUSBCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed