SCHEMBL11024459

SCHEMBL11024459

CCCCCNCC1=CN=C(c2ccccc2)c2ccccc2N1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 2/20 0.39
CCKBR P32239 2/20 0.39
CHRM1 P11229 1/20 0.39
HRH4 Q9H3N8 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
CCNE2 O96020 1/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
SOAT1 P35610 2/20 0.35
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11298881 0.77 CDK2 (0.40) CCKARCCKBRCHRM1HRH4HRH3
SCHEMBL9540291 0.73 HRH4 (0.38) HRH4HRH3SIGMAR1SMN1; SMN2ALDH1A1
SCHEMBL27552511 0.66 GABRA1 (0.48) CCKARCCKBRCHRM1GABRA1GABRG2
Biphenyl SCHEMBL22832517 0.65 SIGMAR1 (0.66) HRH4HRH3SIGMAR1SOAT1ALDH1A1
Biphenyl SCHEMBL5716029 0.65 SIGMAR1 (0.66) HRH4HRH3SIGMAR1SOAT1ALDH1A1
SCHEMBL11032087 0.65 HRH4 (0.38) HRH4HRH3SIGMAR1SOAT1SMN1; SMN2
Biphenyl SCHEMBL27827416 0.64 SIGMAR1 (0.63) HRH4HRH3SIGMAR1SOAT1ALDH1A1
SCHEMBL538475 0.64 MAOA (0.76) HRH4HRH3SIGMAR1SMN1; SMN2MAPT
SCHEMBL1692071 0.62 MAOA (0.80) HRH4HRH3SIGMAR1SMN1; SMN2MEN1
SCHEMBL2882451 0.62 MAOA (0.80) HRH4HRH3SIGMAR1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0054839-B1 2-ACYLAMINOMETHYL-1,4-BENZODIAZEPINES AND THEIR SALTS, METHODS OF PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Kali-Chemie Pharma GmbH (DE) 1985-06-19 EP disclosed
EP-0054839-A2 2-Acylaminomethyl-1,4-benzodiazepines and their salts, methods of preparing them and pharmaceutical compositions containing them Kali-Chemie Pharma GmbH (DE) 1982-06-30 EP disclosed