SCHEMBL11030839

SCHEMBL11030839

O=C1CN(O)CC(CCc2ccccc2)N1C(=O)C1CC1

nearest known ligand 0.41

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SLC18A2 Q05940 1/20 0.40
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11024548 0.94 MTNR1B (0.42) SLC18A2KCNH2
SCHEMBL11026816 0.79 KMT2A (0.46) KCNH2
SCHEMBL11216819 0.76 KMT2A (0.43) KCNH2
SCHEMBL11029433 0.72 SLC18A2 (0.43) SLC18A2KCNH2
SCHEMBL4664890 0.69 MTNR1B (0.40)
SCHEMBL9876918 0.68 SLC18A2 (0.49) SLC18A2
SCHEMBL10994286 0.67 ALDH1A1 (0.55)
SCHEMBL10993438 0.65 HTT (0.45)
SCHEMBL28328103 0.64 ABCB1 (0.60) SLC18A2KCNH2
SCHEMBL14548187 0.63 FAAH (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0086678-B1 PROCESS FOR THE PREPARATION OF 2-ACYL-1,3,4,6,7,11B-2H-HEXAHYDRO-4-PYRAZINO(2,1-A)ISOQUINOLINONES AND INTERMEDIATES ELF SANOFI (FR) 1985-07-03 EP disclosed
EP-0086678-A1 Process for the preparation of 2-acyl-1,3,4,6,7,11b-2H-hexahydro-4-pyrazino(2,1-a)isoquinolinones and intermediates ELF SANOFI (FR) 1983-08-24 EP disclosed