SCHEMBL11039631

SCHEMBL11039631

COC(=O)Oc1nnn(-c2ccc(F)cc2)c1N

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.49
SMN1; SMN2 Q16637 5/20 0.46
PTGS2 P35354 2/20 0.45
NPC1 O15118 4/20 0.42
MAPT P10636 3/20 0.42
LMNA P02545 2/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 3/20 0.41
ALOX15 P16050 1/20 0.41
MAPK14 Q16539 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
IDO1 P14902 2/20 0.40
TDO2 P48775 2/20 0.40
SLC5A1 P13866 1/20 0.39
SLC5A2 P31639 1/20 0.39
GAA P10253 1/20 0.39
GABRA5 P31644 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11038855 0.87 TP53 (0.63) TP53SMN1; SMN2NPC1LMNAHPGD
SCHEMBL11041382 0.86 TP53 (0.49) TP53SMN1; SMN2PTGS2NPC1MAPT
SCHEMBL11044738 0.86 TP53 (0.49) TP53SMN1; SMN2NPC1HPGDRAB9A
SCHEMBL11096860 0.86 SMN1; SMN2 (0.55) TP53SMN1; SMN2LMNAMAPK14NPSR1
SCHEMBL11095871 0.85 TP53 (0.54) TP53SMN1; SMN2LMNAHPGDNPSR1
SCHEMBL11041232 0.82 KMT2A (0.49) TP53SMN1; SMN2NPC1MAPTLMNA
SCHEMBL11040213 0.81 IDO1 (0.43) TP53SMN1; SMN2NPC1MAPTRAB9A
SCHEMBL11044671 0.80 POLB (0.49) TP53SMN1; SMN2MAPTHPGDGAA
SCHEMBL11047507 0.79 MAPT (0.43) TP53SMN1; SMN2NPC1MAPTRAB9A
SCHEMBL10991357 0.78 TP53 (0.74) TP53SMN1; SMN2PTGS2NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0073931-B1 ANILINO-1,2,3-TRIAZOLE DERIVATIVES, MEDICAMENTS CONTAINING THEM, PROCESS FOR PREPARING THEM, AND THEIR USE BOEHRINGER INGELHEIM KG (DE) 1985-02-13 EP disclosed
EP-0073931-A1 Anilino-1,2,3-triazole derivatives, medicaments containing them, process for preparing them, and their use BOEHRINGER INGELHEIM KG (DE) 1983-03-16 EP disclosed