SCHEMBL11040175

SCHEMBL11040175

CS(=O)(=O)O.N#CC(CO)Cc1ccccc1

nearest known ligand 0.47

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.44
CTSK P43235 5/20 0.44
CTSC P53634 4/20 0.43
TRPA1 O75762 1/20 0.43
ANPEP P15144 1/20 0.43
CTSL P07711 6/20 0.43
CTSB P07858 4/20 0.43
CYP3A4 P08684 1/20 0.41
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 1/20 0.40
THRB P10828 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL353200 0.88 TRPA1 (0.48) CTSSCTSKCTSCTRPA1ANPEP
SCHEMBL4426620 0.79 CTSC (0.50) CTSSCTSKCTSCANPEPCYP3A4
SCHEMBL11040202 0.77 ANPEP (0.40) CTSSCTSKCTSCANPEPCTSL
SCHEMBL1343851 0.76 EPHX1 (0.48) CTSSCTSKCTSCANPEPALDH1A1
SCHEMBL11044501 0.75 TRPA1 (0.47) TRPA1CYP3A4MAPK1ALDH1A1THRB
SCHEMBL11044364 0.73 TSHR (0.41) CTSSCTSKTRPA1CTSLCTSB
SCHEMBL14321654 0.73 MAOB (0.42) CTSSCTSKCTSCTRPA1ANPEP
SCHEMBL31118140 0.73 CTSC (0.46) CTSSCTSKCTSCTRPA1
SCHEMBL11020091 0.73 MAOB (0.41) CTSSCTSKCTSCANPEPCTSL
SCHEMBL11045389 0.72 ALDH1A1 (0.44) TRPA1CYP3A4MAPK1ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4490165-A Meta-(phenylalkoxy)phenyl-N-methoxy-N-methylurea compounds, methods for preparing same and herbicidal use thereof AMERICAN CYANAMID COMPANY (US) 1984-12-25 US disclosed
US-4308213-A Meta-(phenylalkoxy)phenyl-N-methoxy-N-methylurea compounds AMERICAN CYANAMID COMPANY (US) 1981-12-29 US disclosed