SCHEMBL11044501

SCHEMBL11044501

CS(=O)(=O)O.OCC(Cl)Cc1ccccc1

nearest known ligand 0.56

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC18A2 known ✓ Q05940 1/20 0.40
TRPA1 O75762 1/20 0.47
CYP3A4 P08684 3/20 0.44
MAPK1 P28482 1/20 0.44
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
GAA P10253 1/20 0.43
BLM P54132 1/20 0.43
GFER P55789 1/20 0.43
PMP22 Q01453 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TSHR P16473 1/20 0.41
CYP1A2 P05177 1/20 0.41
MME P08473 1/20 0.41
TAAR1 Q96RJ0 2/20 0.40
SIGMAR1 Q99720 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9171314 0.87 TRPA1 (0.54) TRPA1TSHRCYP1A2TAAR1SIGMAR1
SCHEMBL7472740 0.87 TRPA1 (0.54) TRPA1TSHRCYP1A2TAAR1SIGMAR1
SCHEMBL11045389 0.76 ALDH1A1 (0.44) TRPA1CYP3A4MAPK1ALDH1A1NPC1
Sulfuric Acid SCHEMBL9718253 0.75 TRPA1 (0.67) TRPA1CYP3A4ALDH1A1KDM4EMAPT
SCHEMBL11040175 0.75 CTSS (0.44) TRPA1CYP3A4MAPK1ALDH1A1NPC1
Benzyl Alcohol SCHEMBL1875625 0.74 TSHR (0.67) CYP3A4ALDH1A1KDM4EMAPTLMNA
Amphetamine SCHEMBL969359 0.74 TAAR1 (0.73) NPC1RAB9ATAAR1SIGMAR1
Amphetamine SCHEMBL973410 0.74 TAAR1 (0.73) NPC1RAB9ATAAR1SIGMAR1
Dextroamphetamine SCHEMBL973408 0.74 TAAR1 (0.73) NPC1RAB9ATAAR1SIGMAR1
Dextroamphetamine SCHEMBL971949 0.74 TAAR1 (0.73) NPC1RAB9ATAAR1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4490165-A Meta-(phenylalkoxy)phenyl-N-methoxy-N-methylurea compounds, methods for preparing same and herbicidal use thereof AMERICAN CYANAMID COMPANY (US) 1984-12-25 US disclosed
US-4308213-A Meta-(phenylalkoxy)phenyl-N-methoxy-N-methylurea compounds AMERICAN CYANAMID COMPANY (US) 1981-12-29 US disclosed