SCHEMBL11043555

SCHEMBL11043555

COC(=O)c1ccc(CCCNCC(O)c2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 8/20 0.48
ADRB2 P07550 3/20 0.48
ADRB3 P13945 7/20 0.46
KDM4E B2RXH2 2/20 0.46
GAA P10253 2/20 0.46
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CYP4A11 Q02928 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11039373 0.94 ADRB1 (0.55) ADRB1ADRB2ADRB3KDM4EGAA
SCHEMBL10731106 0.88 PNMT (0.47) ADRB1ADRB2ADRB3
SCHEMBL6540063 0.87 ADRB1 (0.49) ADRB1ADRB2ADRB3KDM4EGAA
SCHEMBL6540069 0.87 ADRB1 (0.49) ADRB1ADRB2ADRB3KDM4EGAA
SCHEMBL11106888 0.87 ADRB1 (0.44) ADRB1ADRB2ADRB3KDM4EGAA
SCHEMBL10890639 0.86 PNMT (0.48) ADRB1ADRB2KDM4EGAAALDH1A1
SCHEMBL11039327 0.84 ADRB1 (0.48) ADRB1ADRB2ADRB3
SCHEMBL11039896 0.84 ADRB2 (0.47) ADRB1ADRB2ADRB3KDM4EGAA
SCHEMBL11184611 0.84 ADRB3 (0.65) ADRB1ADRB2ADRB3
SCHEMBL11352104 0.83 ADRB1 (0.46) ADRB1ADRB2ADRB3KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0040915-B1 ARYLETHANOLAMINE DERIVATIVES, THEIR PREPARATION AND USE IN PHARMACEUTICAL COMPOSITIONS BEECHAM GROUP PLC (GB) 1984-03-21 EP disclosed
US-4385066-A DIETETICS, HYPERGLYCEMIC AGENTS ANTIINFLAMMATORY AGENTS BEECHAM GROUP LIMITED (GB) 1983-05-24 US disclosed
EP-0040915-A1 Arylethanolamine derivatives, their preparation and use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1981-12-02 EP disclosed